Papers on solid phase organic synthesis published in 1998
This list is arranged by the name of the first author. Any omissions, mistakes and
inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any
reference, please use its ID# -- the last number in the reference.) You are welcome to use this
compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic
database of references in molecular diversity. Internet http://www.5z.com.
Recently added entries are marked in bold
- Anonymous. (1998) Solid phase organic synthesis. J. Chem. Soc. Perkin Trans. 1, v-viii. #10753
- Abraham, S., Rajan, P.K., & Sreekumar, K. (1998) Poly(methyl methacrylate) supported isoxazolinium Cr(VI) species as oxidizing reagents. Ind. J. Chem. B-Org. Chem. Med. Chem., 36B, 769-775. #10775
- Adams, J.H., Cook, R.M., Hudson, D., Jammalamadaka, V., Lyttle, M.H., & Songster, M.F. (1998) A reinvestigation of the preparation, properties, and applications of aminomethyl and 4-methylbenzhydrylamine polystyrene resins. J. Org. Chem., 63, 3706-3716. #12109
- Adinolfi, M., Barone, G., De Napoli, L., Iadonisi, A., & Piccialli, G. (1998) Use of controlled pore glass in solid phase oligosaccharide synthesis. Application to the semiautomated synthesis of a glyconucleotide conjugate. Tetrahedron Lett., 39, 1953-1956. #10614
- Adrian, F.M., Altava, B., Burguete, M.I., Luis, S.V., Salvador, R.V., & Garcia-Espana, E. (1998) Synthetic methods for the preparation of polystyrene resins containing chiral polyamine chains. Tetrahedron, 54, 3581-3588. #12252
- Ajjou, A.N., & Alper, H. (1998) A new, efficient, and in some cases highly regioselective water-soluble polymer rhodium catalyst for olefin hydroformylation. J. Amer. Chem. Soc., 120, 1466-1468. #11797
- Akerblom, E.B., Nygren, A.S., & Agback, K.H. (1998) Six new photolabile linkers for solid-phase synthesis. 1. Methods of preparation. Mol. Diversity, 3, 137-148. #10881
- Albert, R., Knecht, H., Andersen, E., Hungerford, V., Schreier, M.H., & Papageorgiou, C. (1998) Isoxazolylthioamides as potential immunosuppressants a combinatorial chemistry approach. Bioorg. Med. Chem. Lett., 8, 2203-2208. #11187
- Aldrian-Herrada, G., Rabie, A., Wintersteiger, R., & Brugidou, J. (1998) Solid-phase synthesis of peptide nucleic acid (PNA) monomers and their oligomerization using disulphide anchoring linkers. J. Peptide Sci., 4, 266-281. #10878
- Allanson, N.M., Liu, D., Chi, F., Jain, R.K., Chen, A., Ghosh, M., Hong, L., & Sofia, M.J. (1998) Synthesis of phenyl 1-thioglycopyranosiduronic acids using a sonicated Jones oxidation. Tetrahedron Lett., 39, 1889-1892. #10612
- Alsina, J., Rabanal, F., Chiva, C., Giralt, E., & Albericio, F. (1998) Active carbonate resins: Application to the solid-phase synthesis of alcohol, carbamate and cyclic peptides. Tetrahedron, 54, 10125-10152. #11248
- Alvarez, K., Tworkowski, I., Vasseur, J.J., Imbach, J.L., & Rayner, B. (1998) A reinvestigation of sulfenyl groups as amino protecting groups for the synthesis of oligonucleotides on solid support by phosphoramidite chemistry. Nucleosides Nucleotides, 17, 365-378. #12201
- Andersen, J.A.M., Karodia, N., Miller, D.J., Stones, D., & Gani, D. (1998) Preparation and catalytic properties of resin bound binuclear rhodium tetracarboxylate complexes. Tetrahedron Lett., 39, 7815-7818. #11585
- Anderson, E.M., Karin, M., & Kirk, O. (1998) One biocatalyst - many applications: The use of Candida antarctica B-lipase in organic synthesis. Biocatalysis and Biotransformation, 16, 181-204. #12302
- Andres, C.J., Swann, R.T., Severino, J., Grant-Young, K., Edinger, K., Mongillo, J., & Deshpande, M.S. (1998) A novel parallel distributor for dispensing of Irori(TM) Rf-encoded tags to microkans in 96-well format. Biotech. Bioeng. (Comb. Chem. ), 61, 93-94. #11250
- Andres, C.J., Whitehouse, D.L., & Deshpande, M.S. (1998) Transition-metal-mediated reactions in combinatorial synthesis. Curr. Opin. Chem. Biol., 2, 353-362. #12073
- Anne, C., Fournie-Zaluski, M.C., Roques, B.P., & Cornille, F. (1998) Solid phase synthesis of peptoid derivatives containing a free C-terminal carboxylate. Tetrahedron Lett., 39, 8973-8974. #11941
- Aronov, A.M., & Gelb, M.H. (1998) Phthalimide resin reagent for efficient Mitsunobu amino-dehydroxylation. Tetrahedron Lett., 39, 4947-4950. #11159
- Arsequell, G., Espuna, G., Valencia, G., Barluenga, J., Perez Carlon, R., & Gonzalez, J.M. (1998) First aromatic electrophilic iodination reaction on the solid-phase: Iodination of bioactive peptides. Tetrahedron Lett., 39, 7393-7396. #11574
- Asseline, U., Roig, V., & Thuong, N.T. (1998) Modified oligonucleotides with a 5'-5' interbase semi-rigid junction for alternate strand triplex formation. Tetrahedron Lett., 39, 8991-8994. #11942
- Avdagic, A., & Sunjic, V. (1998) Biocatalytic deracemization of 1,4-benzodiazepines in the synthesis of enantiomerically pure serine. Helv. Chim. Acta, 81, 85-92. #10684
- Baker, C.T., Salituro, F.G., Court, J.J., Deininger, D.D., Kim, E.E., Li, B.Q., Novak, P.M., Rao, B.G., Pazhanisamy, S., Schairer, W.C., & Tung, R.D. (1998) Design, synthesis, and conformational analysis of a novel series of HIV protease inhibitors. Bioorg. Med. Chem. Lett., 8, 3631-3636. #12305
- Baldwin, J.J. (1998) Small molecule libraries: Overview of issues and strategies in library design. In E.M. Gordon & J.F.J. Kerwin (Eds.), Combinatorial Chemistry and Molecular Diversity in Drug Discovery. (pp. 181-188). John Wiley & Sons, New York. #11711
- Ball, C.P., Barrett, A.G.M., Commercon, A., Compere, D., Kuhn, C., Roberts, R.S., Smith, M.L., & Venier, O. (1998) Chameleon catches in combinatorial chemistry: Tebbe olefination of polymer supported esters and the synthesis of amines, cyclohexanones, enones, methyl ketones and thiazoles. Chem. Commun., 2019-2020. #11821
- Ball, C.P., Barrett, A.G.M., Poitout, L.F., Smith, M.L., & Thorn, Z.E. (1998) Polymer backbone disassembly: Polymerisable templates and vanishing supports in high loading parallel synthesis. Chem. Commun., 2453-2454. #12110
- Baraniak, J., Korczynski, D., Kaczmarek, R., & Wasilewska, E. (1998) New approach to the solid phase synthesis of N3'->P5' phosphoramidate oligonucleotides. Nucleosides Nucleotides, 17, 1347-1353. #11252
- Barawkar, D.A., Linkletter, B., & Bruice, T.C. (1998) Synthesis of protected guanidinium linked dinucleoside incorporable into an oligonucleotide using solid phase DNA methodology. Bioorg. Med. Chem. Lett., 8, 1517-1520. #11191
- Barawkar, D.A., & Bruice, T.C. (1998) Synthesis, biophysical properties, and nuclease resistance properties of mixed backbone oligodeoxynucleotides containing cationic internucleoside guanidinium linkages: Deoxynucleic guanidine/DNA chimeras. Proc. Natl. Acad. Sci. USA, 95, 11047-11052. #11185
- Barbaste, M., Rolland-Fulcrand, V., Roumestant, M.L., Viallefont, P., & Martinez, J. (1998) Rapid solid phase synthesis of alpha-amino acids. Tetrahedron Lett., 39, 6287-6290. #11026
- Barco, A., Benetti, S., De Risi, C., Marchetti, P., Pollini, G.P., & Zanirato, V. (1998) Polymer-bound 4-benzyl-sulfonyl-1-triphenylphosphoranylidene-2-butanone as a tool for the solid-phase synthesis of substituted piperidin-4-one derivatives. Tetrahedron Lett., 39, 7591-7594. #11565
- Barlaam, B., Hamon, A., & Maudet, M. (1998) New hydroxylamines for the synthesis of hydroxamic acids. Tetrahedron Lett., 39, 7865-7868. #11822
- Bauser, M., Winter, M., Valenti, C.A., Wiesmuller, K.H., & Jung, G. (1998) Synthesis of hydantoins via N,N'-ureas derived from polymer-bound amino acids. Mol. Diversity, 3, 257-260. #12101
- Baxter, E.W., Rueter, J.K., Nortey, S.O., & Reitz, A.B. (1998) Arylsulfonate esters in solid phase organic synthesis. II.Compatibility with commonly-used reaction conditions. Tetrahedron Lett., 39, 979-982. #10491
- Becker, H.F., Grosjean, H., & Fourrey, J.L. (1998) Chemical synthesis of 4-thiouridine-containing substrate analogues of tRNA : Pseudouridine-55 synthase: Photocross-linking studies. Nucleosides Nucleotides, 17, 2403-2416. #12309
- Beltran, M., Pedroso, E., & Grandas, A. (1998) A comparison of histidine protecting groups in the synthesis of peptide-oligonucleotide conjugates. Tetrahedron Lett., 39, 4115-4118. #10841
- Bender, D., & Gee, A.D. (1998) Solid phase-supported reaction of N.C.A.H11CN with arabinose: A simplified automated synthesis of D-[1-11C]glucose. J. Label. Compound. Radiopharm., 41, 287-300. #10757
- Bengtsson, M., Broddefalk, J., Dahmen, J., Henriksson, K., Kihlberg, J., Lonn, H., Srinivasa, B.R., & Stenvall, K. (1998) Convergent synthesis of neoglycopeptides by coupling of 2-bromoethyl glycosides to cysteine and homocysteine residues in T cell stimulating peptides. Glycoconjugate J., 15, 223-231. #10703
- Berlin, K., Jain, R.K., Simon, M.D., & Richert, C. (1998) A porphyrin embedded in DNA. J. Org. Chem., 63, 1527-1535. #10780
- Berteina, S., Wendeborn, S., & De Mesmaeker, A. (1998) Radical and palladium-mediated cyclizations of ortho-iodo benzyl enamines: Application to solid phase synthesis. Synlett, 1231. #12310
- Berteina, S., & De Mesmaeker, A. (1998) Application of radical chemistry to solid support synthesis. Tetrahedron Lett., 39, 5759-5762. #10965
- Bertini, V., Lucchesini, F., Pocci, M., & De Munno, A. (1998) 1,3-Dithiane polymers for the supported synthesis of ketones. Tetrahedron Lett., 39, 9263-9266. #12019
- Beutel, B.A. (1998) Strategies for screening combinatorial libraries. In E.M. Gordon & J.F.J. Kerwin (Eds.), Combinatorial Chemistry and Molecular Diversity in Drug Discovery. (pp. 421-432). John Wiley & Sons, New York. #11727
- Bhalay, G., & Dunstan, A.R. (1998) Facile solid phase synthesis of an activated diazo linker. Tetrahedron Lett., 39, 7803-7806. #11577
- Bhalay, G., Cowell, D., Hone, N.D., Scobie, M., & Baxter, A.D. (1998) Multiple solid-phase synthesis of hydantoins and thiohydantoins. Mol. Diversity, 3, 195-198. #11255
- Bhandari, A., Jones, D.G., Schullek, J.R., Vo, K., Schunk, C.A., Tamanaha, L.L., Chen, D., Yuan, Z., Needels, M.C., & Gallop, M.A. (1998) Exploring structure-activity relationship around the phosphomannose isomerase inhibitor AF14049 via combinatorial synthesis. Bioorg. Med. Chem. Lett., 8, 2303-2308. #11198
- Bianco, A., Zabel, C., Walden, P., & Jung, G. (1998) N-hydroxy-amide analogues of MHC-class I peptide ligands with nanomolar binding affinities. J. Peptide Sci., 4, 471-478. #12313
- Bicknell, A.J., Hird, N.W., & Readshaw, S.A. (1998) Efficient robotic synthesis. Multi-component preparation of a tricyclic template by solid phase Tsuge reaction. Tetrahedron Lett., 39, 5869-5872. #10968
- Bienayme, H., & Bouzid, K. (1998) Synthesis of rigid hydrophobic tetrazoles using an Ugi multi-component heterocyclic condensation. Tetrahedron Lett., 39, 2735-2738. #10748
- Bilodeau, M.T., & Cunningham, A.M. (1998) Solid-supported synthesis of imidazoles: A strategy for direct resin-attachment to the imidazole core. J. Org. Chem., 63, 2800-2801. #10754
- Bing, Y. (1998) Monitoring the progress and the yield of solid-phase organic reactions directly on resin supports. Account. Chem. Res., 31, 621-630. #12219
- Blackburn, C. (1998) Polymer supports for solid-phase organic synthesis. Biopolymers (Pept. Sci. ), 47, 311-351. #12261
- Blackburn, C. (1998) A three-component solid-phase synthesis of 3-aminoimidazol[1,2-a]azines. Tetrahedron Lett., 39, 5469-5472. #10954
- Blaskovich, M.A., & Kahn, M. (1998) Polymer-supported acetylide addition to hexa-2,4-dienal. Synthesis-Stuttgart, 965-966. #12236
- Blaskovich, M.A., & Kahn, M. (1998) Solid-phase preparation of dienes. J. Org. Chem., 63, 1119-1125. #11798
- Bleczinski, C.F., & Richert, C. (1998) Monitoring the hybridization of the components of oligonucleotide mixtures to immobilized DNA via matrix-assisted laser desorption/ionization time-of-flight mass spectrometry. Rapid Commun. Mass Spectrom., 12, 1737-1743. #12315
- Bleicher, K.H., & Wareing, J.R. (1998) PhFl polystyrene: A new resin for solid phase organic synthesis. Tetrahedron Lett., 39, 4587-4590. #11171
- Bleicher, K.H., & Wareing, J.R. (1998) PhFl acetic acid: A new linker for solid phase organic synthesis. Tetrahedron Lett., 39, 4591-4594. #11164
- Blixt, O., & Norberg, T. (1998) Solid-phase enzymatic synthesis of a sialyl Lewis x tetrasaccharide on a sepharose matrix. J. Org. Chem., 63, 2705-2710. #10994
- Boeijen, A., Kruijtzer, J.A.W., & Liskamp, R.M.J. (1998) Combinatorial chemistry of hydantoins. Bioorg. Med. Chem. Lett., 8, 2375-2380. #11210
- Bogdan, F.M., & Chow, C.S. (1998) The synthesis of allyl- and allyloxycarbonyl-protected RNA phosphoramidites. Useful reagents for solid-phase synthesis of RNAs with base-labile modifications. Tetrahedron Lett., 39, 1897-1900. #10613
- Boger, D.L., Goldberg, J., Jiang, W.Q., Chai, W.Y., Ducray, P., Lee, J.K., Ozer, R.S., & Andersson, C.M. (1998) Higher order iminodiacetic acid libraries for probing protein-protein interactions. Bioorg. Med. Chem., 6, 1347-1378. #11825
- Bohm, G., Dowden, J., Rice, D.C., Burgess, I., Pilard, J.F., Guilbert, B., Haxton, A., Hunter, R.C., Turner, N.J., & Flitsch, S.L. (1998) A novel linker for the attachment of alcohols to solid supports. Tetrahedron Lett., 39, 3819-3822. #10849
- Bondy, S.S. (1998) The role of automation in drug discovery. Curr. Opin. Drug. Disc. Develop., 1, 116-119. #11395
- Booth, S., Hermkens, P.H.H., Ottenheijm, H.C.J., & Rees, D.C. (1998) Solid-phase organic reactions III: A review of the literature Nov 96-Dec 97. Tetrahedron, 54, 15385-15443. #12237
- Boussie, T.R., Coutard, C., Turner, H., Murphy, V., & Powers, T.S. (1998) Solid-phase synthesis and encoding strategies for olefin polymerization catalyst libraries. Angew. Chem. Int. Ed., 37, 3272-3275. #12139
- Boymond, L., Rottlander, M., Cahiez, G., & Knochel, P. (1998) Preparation of highly functionalized Grignard reagents by an iodine-magnesium exchange reaction and its application in solid-phase synthesis. Angew. Chem. Int. Ed., 37, 1701-1703. #11257
- Brady, S.F., Stauffer, K.J., Lumma, W.C., Smith, G.M., Ramjit, H.G., Lewis, S.D., Lucas, B.J., Gardell, S.J., Lyle, E.A., Appleby, S.D., Cook, J.J., Holahan, M.A., Stranieri, M.T., Lynch, J.J.Jr., Lin, J.H., Chen, I.W., Vastag, K., Naylor-Olsen, A.M., & Vacca, J.P. (1998) Discovery and development of the novel potent orally active thrombin inhibitor N-(9-hydroxy-9-fluorenecar-boxy)prolyl trans-4-aminocyclohexylmethyl amide (L-372,460): Coapplication of structure-based design and rapid multiple analogue synthesis on solid support. J. Med. Chem., 41, 401-406. #11236
- Bray, A.M., Maeji, N.J., Lagniton, L.M., Chiefari, D., James, I.W., Ang, K., Ede, N., Valerio, R.M. & Mason, T.J. (1998) Simultaneous multiple synthesis by the Multipin(TM) method: Techniques for multiple handling,high throughput characterization and reaction optimization on solid phase. In X. Xu, Y. Ye & J.P. Tam (Eds.), Peptides. Biology and Chemistry. Proceedings of the 1996 Chinese Peptide Symposium. (pp. 67. Kluwer/ESCOM, Dordrecht. #14303
- Breitenbucher, J.G., Johnson, C.R., Haight, M., & Phelan, J.C. (1998) Generation of a piperazine-2-carboxamide library: A practical application of the phenol-sulfide react and release linker. Tetrahedron Lett., 39, 1295-1298. #10510
- Breitenbucher, J.G., & Hui, H.C. (1998) Titanium mediated reductive amination on solid support: Extending the utility of the 4-hydroxy-thiophenol linker. Tetrahedron Lett., 39, 8207-8210. #12009
- Brennan, T., Biddison, G., Frauendorf, A., Schwarcz, L., Keen, B., Ecker, D.J., Davis, P.W., Tinder, R., & Swayze, E.E. (1998) Two-dimensional parallel array technology as a new approach to automated combinatorial solid-phase organic synthesis. Biotech. Bioeng. (Comb. Chem. ), 61, 33-45. #10759
- Breslow, R. (1998) Bioorganic chemistry: A natural and unnatural science. J. Chem. Educ., 75, 705-718. #10970
- Brill, W.K.D., De Mesmaeker, A., & Wendeborn, S. (1998) Solid phase synthesis of levoglucosan derivatives. Synlett, 1085-1090. #12318
- Brill, W.K.D., Schmidt, E., & Tommasi, R.A. (1998) Immobilizations of nucleophiles on polystyrene supports. Synlett, 906. #11258
- Broddefalk, J., Bergquist, K.E., & Kihlberg, J. (1998) Use of acid-labile protective groups for carbohydrate moieties in synthesis of glycopeptides related to type II collagen. Tetrahedron, 54, 12047-12070. #11828
- Brown, D.S., Revill, J.M., & Shute, R.E. (1998) Merrifield, alpha-methoxyphenyl (MAMP) resin: A new versatile solid support for the synthesis of secondary amides. Tetrahedron Lett., 39, 8533-8536. #11946
- Brown, R.C.D. (1998) Recent developments in solid-phase organic synthesis. J. Chem. Soc. Perkin Trans. 1, 3293-3320. #11829
- Buchardt, J., & Meldal, M. (1998) A chemically inert hydrophilic resin for solid phase organic synthesis. Tetrahedron Lett., 39, 8695-8698. #11962
- Buchstaller, H.P. (1998) Solid phase synthesis of oxazolidinones via a novel cyclisation/cleavage reaction. Tetrahedron, 54, 3465-3470. #11050
- Bui, C.T., Rasoul, F.A., Ercole, F., Pham, Y., & Maeji, N.J. (1998) Efficiencies of reductive amination reactions on different solid supports. Tetrahedron Lett., 39, 9279-9282. #12020
- Bunin, B.A. (1998) The Combinatorial Index. Academic Press, San Diego. ISBN 0121413403 #10496
- Burke, T.R., & Zhang, Z.Y. (1998) Protein-tyrosine phosphatases: Structure, mechanism, and inhibitor discovery. Biopolymers, 47, 225-241. #12323
- Butenandt, J., Eker, A.P.M., & Carell, T. (1998) Synthesis, crystal structure, and enzymatic evaluation of a DNA-photolesion isostere. Chem. Eur. J., 4, 642-654. #10991
- Byk, G., Dubertret, C., Escriou, V., Frederic, M., Jaslin, G., Rangara, R., Pitard, B., Crouzet, J., Wils, P., Schwartz, B., & Scherman, D. (1998) Synthesis, activity, and structure-activity relationship studies of novel cationic lipids for DNA transfer. J. Med. Chem., 41, 224-235. #10751
- Byk, G., Soto, J., Mattler, C., Frederic, M., & Scherman, D. (1998) Novel non-viral vectors for gene delivery: Synthesis of a second-generation library of mono-functionalized poly-(guanidinium)amines and their introduction into cationic lipids. Biotechnol. Bioeng., 61, 81-87. #12221
- Campian, E., Peterson, M.L., Saneii, H.H., & Furka, A. (1998) Deconvolution by omission libraries. Bioorg. Med. Chem. Lett., 8, 2357-2362. #11207
- Cano, M., Camps, F., & Joglar, J. (1998) Solid phase synthesis of cyclopropenes. Tetrahedron Lett., 39, 9819-9822. #12044
- Cao, J., Cuny, G.D., & Hauske, J.R. (1998) Ring opening cross-metathesis on solid support: A combinatorial library synthesis of highly functionalized cyclopentanes. Mol. Diversity, 3, 173-179. #10884
- Cao, L.Q., Bornscheuer, U.T., & Schmid, R.D. (1998) Lipase-catalyzed solid-phase synthesis of sugar esters. IV. Selectivity of lipases towards primary and secondary hydroxyl groups in carbohydrates. Biocatalysis and Biotransformation, 16, 249-257. #12324
- Carroll, C.D., Patel, H., Johnson, T.O., Guo, T., Orlowski, M., He, Z.M., Cavallaro, C.L., Guo, J., Oksman, A., Gluzman, I.Y., Connelly, J., Chelsky, D., Goldberg, D.E., & Dolle, R.E. (1998) Identification of potent inhibitors of Plasmodium falciparum plasmepsin II from an encoded statine combinatorial library. Bioorg. Med. Chem. Lett., 8, 2315-2320. #11200
- Casebier, D., & Baldino, C. (1998) Advances in combinatorial chemistry. Innovations in Pharmaceutical Technology, 1, 63-67. #12089
- Chaix, C., Minard-Basquin, C., Delair, T., Pichot, C., & Mandrand, B. (1998) Oligonucleotide synthesis on maleic anhydride copolymers covalently bound to silica spherical support and characterization of the obtained conjugates. J. Appl. Polym. Sci., 70, 2487-2497. #12327
- Chamoin, S., Houldsworth, S., & Snieckus, V. (1998) The Stille cross coupling reactions on solid support. Link to solution phase directed ortho metalation. An ester linker approach to styryl, biaryl and heterobiaryl carboxylic acids. Tetrahedron Lett., 39, 4175-4178. #10854
- Chamoin, S., Houldsworth, S., Kruse, C.G., Bakker, I., & Snieckus, V. (1998) The Suzuki-Miyaura cross coupling reactions on solid support. Link to solution phase directed ortho metalation. The Leznoff acetal linker approach to biaryl and heterobiaryl aldehydes. Tetrahedron Lett., 39, 4179-4182. #10855
- Chandrasekhar, S., & Padmaja, M.B. (1998) Practical preparation of first carbon linked polymer bound 1,3-diol. Syn. Commun., 28, 3715-3720. #11834
- Chen, C., McDonald, I.A., & Munoz, B. (1998) Synthesis of dihydropyridone scaffolds on solid support: Resin Activation/Capture Approach/REACAP Technology. Tetrahedron Lett., 39, 217-220. #9869
- Chen, C., & Munoz, B. (1998) Solid phase synthesis of 2,4-disubstituted pyridine and tetrahydropyridine derivatives: Resin activation/capture approach/REACAP technology. Tetrahedron Lett., 39, 3401-3404. #10805
- Chen, C., & Munoz, B. (1998) Solid phase synthesis of N-acyl-2-substituted-dihydro-4-pyridone: Resin activation/capture approach/REACAP technology. Tetrahedron Lett., 39, 6781-6784. #11224
- Chen, S., & Janda, K.D. (1998) Total synthesis of naturally occuring prostaglandin F(2alpha) on a non-cross-linked polystyrene support. Tetrahedron Lett., 39, 3943-3946. #10840
- Chen, X.T., Sames, D., & Danishefsky, S.J. (1998) Exploration of modalities in building alpha-O-linked systems through glycal assembly: A total synthesis of the mucin-related F1-alpha antigen. J. Amer. Chem. Soc., 120, 7760-7769. #11265
- Cheng, J.F., & Mjalli, A.M.M. (1998) Solid-phase synthesis of D2-isoxazolines. Tetrahedron Lett., 39, 939-942. #10488
- Chhabra, S.R., Khan, A.N., & Bycroft, B.W. (1998) Versatile Dde-based primary amine linkers for solid phase synthesis. Tetrahedron Lett., 39, 3585-3588. #10809
- Chin, J., Fell, B., Pochapsky, S., Shapiro, M.J., & Wareing, J.R. (1998) 2D SECSY NMR for combinatorial chemistry: High-resolution MAS spectra for resin-bound molecules. J. Org. Chem., 63, 1309-1311. #10664
- Cho, C.Y., Youngquist, R.S., Paikoff, S.J., Beresini, M.H., Hebert, A.R., Berleau, L.T., Liu, C.W., Wemmer, D.E., Keough, T., & Schultz, P.G. (1998) Synthesis and screening of linear and cyclic oligocarbamate libraries: Discovery of high affinity ligands for GPIIb/IIIa. J. Amer. Chem. Soc., 120, 7706-7718. #11266
- Chou, Y.L., Morrissey, M.M., & Mohan, R. (1998) Novel serine-based linker for the solid-phase synthesis of organic compounds. Tetrahedron Lett., 39, 757-760. #10050
- Christopher, J., & Lea, L. (1998) Perkin 1 abstracts: Solid phase organic synthesis. J. Chem. Soc. Perkin Trans. 1, vii-x. #11016
- Collins, J.L., Blanchard, S.G., Boswell, G.E., Charifson, P.S., Cobb, J.E., Henke, B.R., Hull-Ryde, E.A., Kazmierski, W.M., Lake, D.H., Leesnitzer, L.M., Lehmann, J., Lenhard, J.M., Orband-Miller, L.A., Gray-Nunez, Y., Parks, D.J., Plunkett, K.D., & Tong, W.Q. (1998) N-(2-benzoylphenyl)-L-tyrosine PPAR gamma agonists. 2. Structure-activity relationship and optimization of the phenyl alkyl ether moiety. J. Med. Chem., 41, 5037-5054. #12335
- Conroy, J.L., Abato, P., Ghosh, M., Austermuhle, M.I., Kiefer, M.R., & Seto, C.T. (1998) Synthesis of cyclohexanone-based cathepsin B inhibitors that interact with both the S and S' binding sites. Tetrahedron Lett., 39, 8253-8256. #12013
- Coppola, G.M. (1998) A new scavenger resin for amines. Tetrahedron Lett., 39, 8233-8236. #12011
- Corbett, J.W. (1998) Recent progress in solid phase heterocycle syntheses. A review. Organic Preparations and Procedures International, 30, 489-550. #14225
- Cornille, F., Emery, P., Schuler, W., Lenoir, C., Mach, B., Rogues, B.P., & Reith, W. (1998) DNA binding properties of a chemically synthesized DNA binding domain of hRFX1. Nucl. Acid. Res., 26, 2143-2149. #11110
- Craig, D., Robson, M.J., & Shaw, S.J. (1998) Traceless linkers for solid-phase synthesis. Homo- and hetero-Diels-Alder reactions of o-quinodimethanes. Synlett, 1381-1383. #12336
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