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Papers on solid phase organic synthesis published in 1998

This list is arranged by the name of the first author. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.


Recently added entries are marked in bold

  1. Anonymous. (1998) Solid phase organic synthesis. J. Chem. Soc. Perkin Trans. 1, v-viii. #10753

  2. Abraham, S., Rajan, P.K., & Sreekumar, K. (1998) Poly(methyl methacrylate) supported isoxazolinium Cr(VI) species as oxidizing reagents. Ind. J. Chem. B-Org. Chem. Med. Chem., 36B, 769-775. #10775

  3. Adams, J.H., Cook, R.M., Hudson, D., Jammalamadaka, V., Lyttle, M.H., & Songster, M.F. (1998) A reinvestigation of the preparation, properties, and applications of aminomethyl and 4-methylbenzhydrylamine polystyrene resins. J. Org. Chem., 63, 3706-3716. #12109

  4. Adinolfi, M., Barone, G., De Napoli, L., Iadonisi, A., & Piccialli, G. (1998) Use of controlled pore glass in solid phase oligosaccharide synthesis. Application to the semiautomated synthesis of a glyconucleotide conjugate. Tetrahedron Lett., 39, 1953-1956. #10614

  5. Adrian, F.M., Altava, B., Burguete, M.I., Luis, S.V., Salvador, R.V., & Garcia-Espana, E. (1998) Synthetic methods for the preparation of polystyrene resins containing chiral polyamine chains. Tetrahedron, 54, 3581-3588. #12252

  6. Ajjou, A.N., & Alper, H. (1998) A new, efficient, and in some cases highly regioselective water-soluble polymer rhodium catalyst for olefin hydroformylation. J. Amer. Chem. Soc., 120, 1466-1468. #11797

  7. Akerblom, E.B., Nygren, A.S., & Agback, K.H. (1998) Six new photolabile linkers for solid-phase synthesis. 1. Methods of preparation. Mol. Diversity, 3, 137-148. #10881

  8. Albert, R., Knecht, H., Andersen, E., Hungerford, V., Schreier, M.H., & Papageorgiou, C. (1998) Isoxazolylthioamides as potential immunosuppressants a combinatorial chemistry approach. Bioorg. Med. Chem. Lett., 8, 2203-2208. #11187

  9. Aldrian-Herrada, G., Rabie, A., Wintersteiger, R., & Brugidou, J. (1998) Solid-phase synthesis of peptide nucleic acid (PNA) monomers and their oligomerization using disulphide anchoring linkers. J. Peptide Sci., 4, 266-281. #10878

  10. Allanson, N.M., Liu, D., Chi, F., Jain, R.K., Chen, A., Ghosh, M., Hong, L., & Sofia, M.J. (1998) Synthesis of phenyl 1-thioglycopyranosiduronic acids using a sonicated Jones oxidation. Tetrahedron Lett., 39, 1889-1892. #10612

  11. Alsina, J., Rabanal, F., Chiva, C., Giralt, E., & Albericio, F. (1998) Active carbonate resins: Application to the solid-phase synthesis of alcohol, carbamate and cyclic peptides. Tetrahedron, 54, 10125-10152. #11248

  12. Alvarez, K., Tworkowski, I., Vasseur, J.J., Imbach, J.L., & Rayner, B. (1998) A reinvestigation of sulfenyl groups as amino protecting groups for the synthesis of oligonucleotides on solid support by phosphoramidite chemistry. Nucleosides Nucleotides, 17, 365-378. #12201

  13. Andersen, J.A.M., Karodia, N., Miller, D.J., Stones, D., & Gani, D. (1998) Preparation and catalytic properties of resin bound binuclear rhodium tetracarboxylate complexes. Tetrahedron Lett., 39, 7815-7818. #11585

  14. Anderson, E.M., Karin, M., & Kirk, O. (1998) One biocatalyst - many applications: The use of Candida antarctica B-lipase in organic synthesis. Biocatalysis and Biotransformation, 16, 181-204. #12302

  15. Andres, C.J., Swann, R.T., Severino, J., Grant-Young, K., Edinger, K., Mongillo, J., & Deshpande, M.S. (1998) A novel parallel distributor for dispensing of Irori(TM) Rf-encoded tags to microkans in 96-well format. Biotech. Bioeng. (Comb. Chem. ), 61, 93-94. #11250

  16. Andres, C.J., Whitehouse, D.L., & Deshpande, M.S. (1998) Transition-metal-mediated reactions in combinatorial synthesis. Curr. Opin. Chem. Biol., 2, 353-362. #12073

  17. Anne, C., Fournie-Zaluski, M.C., Roques, B.P., & Cornille, F. (1998) Solid phase synthesis of peptoid derivatives containing a free C-terminal carboxylate. Tetrahedron Lett., 39, 8973-8974. #11941

  18. Aronov, A.M., & Gelb, M.H. (1998) Phthalimide resin reagent for efficient Mitsunobu amino-dehydroxylation. Tetrahedron Lett., 39, 4947-4950. #11159

  19. Arsequell, G., Espuna, G., Valencia, G., Barluenga, J., Perez Carlon, R., & Gonzalez, J.M. (1998) First aromatic electrophilic iodination reaction on the solid-phase: Iodination of bioactive peptides. Tetrahedron Lett., 39, 7393-7396. #11574

  20. Asseline, U., Roig, V., & Thuong, N.T. (1998) Modified oligonucleotides with a 5'-5' interbase semi-rigid junction for alternate strand triplex formation. Tetrahedron Lett., 39, 8991-8994. #11942

  21. Avdagic, A., & Sunjic, V. (1998) Biocatalytic deracemization of 1,4-benzodiazepines in the synthesis of enantiomerically pure serine. Helv. Chim. Acta, 81, 85-92. #10684

  22. Baker, C.T., Salituro, F.G., Court, J.J., Deininger, D.D., Kim, E.E., Li, B.Q., Novak, P.M., Rao, B.G., Pazhanisamy, S., Schairer, W.C., & Tung, R.D. (1998) Design, synthesis, and conformational analysis of a novel series of HIV protease inhibitors. Bioorg. Med. Chem. Lett., 8, 3631-3636. #12305

  23. Baldwin, J.J. (1998) Small molecule libraries: Overview of issues and strategies in library design. In E.M. Gordon & J.F.J. Kerwin (Eds.), Combinatorial Chemistry and Molecular Diversity in Drug Discovery. (pp. 181-188). John Wiley & Sons, New York. #11711

  24. Ball, C.P., Barrett, A.G.M., Commercon, A., Compere, D., Kuhn, C., Roberts, R.S., Smith, M.L., & Venier, O. (1998) Chameleon catches in combinatorial chemistry: Tebbe olefination of polymer supported esters and the synthesis of amines, cyclohexanones, enones, methyl ketones and thiazoles. Chem. Commun., 2019-2020. #11821

  25. Ball, C.P., Barrett, A.G.M., Poitout, L.F., Smith, M.L., & Thorn, Z.E. (1998) Polymer backbone disassembly: Polymerisable templates and vanishing supports in high loading parallel synthesis. Chem. Commun., 2453-2454. #12110

  26. Baraniak, J., Korczynski, D., Kaczmarek, R., & Wasilewska, E. (1998) New approach to the solid phase synthesis of N3'->P5' phosphoramidate oligonucleotides. Nucleosides Nucleotides, 17, 1347-1353. #11252

  27. Barawkar, D.A., Linkletter, B., & Bruice, T.C. (1998) Synthesis of protected guanidinium linked dinucleoside incorporable into an oligonucleotide using solid phase DNA methodology. Bioorg. Med. Chem. Lett., 8, 1517-1520. #11191

  28. Barawkar, D.A., & Bruice, T.C. (1998) Synthesis, biophysical properties, and nuclease resistance properties of mixed backbone oligodeoxynucleotides containing cationic internucleoside guanidinium linkages: Deoxynucleic guanidine/DNA chimeras. Proc. Natl. Acad. Sci. USA, 95, 11047-11052. #11185

  29. Barbaste, M., Rolland-Fulcrand, V., Roumestant, M.L., Viallefont, P., & Martinez, J. (1998) Rapid solid phase synthesis of alpha-amino acids. Tetrahedron Lett., 39, 6287-6290. #11026

  30. Barco, A., Benetti, S., De Risi, C., Marchetti, P., Pollini, G.P., & Zanirato, V. (1998) Polymer-bound 4-benzyl-sulfonyl-1-triphenylphosphoranylidene-2-butanone as a tool for the solid-phase synthesis of substituted piperidin-4-one derivatives. Tetrahedron Lett., 39, 7591-7594. #11565

  31. Barlaam, B., Hamon, A., & Maudet, M. (1998) New hydroxylamines for the synthesis of hydroxamic acids. Tetrahedron Lett., 39, 7865-7868. #11822

  32. Bauser, M., Winter, M., Valenti, C.A., Wiesmuller, K.H., & Jung, G. (1998) Synthesis of hydantoins via N,N'-ureas derived from polymer-bound amino acids. Mol. Diversity, 3, 257-260. #12101

  33. Baxter, E.W., Rueter, J.K., Nortey, S.O., & Reitz, A.B. (1998) Arylsulfonate esters in solid phase organic synthesis. II.Compatibility with commonly-used reaction conditions. Tetrahedron Lett., 39, 979-982. #10491

  34. Becker, H.F., Grosjean, H., & Fourrey, J.L. (1998) Chemical synthesis of 4-thiouridine-containing substrate analogues of tRNA : Pseudouridine-55 synthase: Photocross-linking studies. Nucleosides Nucleotides, 17, 2403-2416. #12309

  35. Beltran, M., Pedroso, E., & Grandas, A. (1998) A comparison of histidine protecting groups in the synthesis of peptide-oligonucleotide conjugates. Tetrahedron Lett., 39, 4115-4118. #10841

  36. Bender, D., & Gee, A.D. (1998) Solid phase-supported reaction of N.C.A.H11CN with arabinose: A simplified automated synthesis of D-[1-11C]glucose. J. Label. Compound. Radiopharm., 41, 287-300. #10757

  37. Bengtsson, M., Broddefalk, J., Dahmen, J., Henriksson, K., Kihlberg, J., Lonn, H., Srinivasa, B.R., & Stenvall, K. (1998) Convergent synthesis of neoglycopeptides by coupling of 2-bromoethyl glycosides to cysteine and homocysteine residues in T cell stimulating peptides. Glycoconjugate J., 15, 223-231. #10703

  38. Berlin, K., Jain, R.K., Simon, M.D., & Richert, C. (1998) A porphyrin embedded in DNA. J. Org. Chem., 63, 1527-1535. #10780

  39. Berteina, S., Wendeborn, S., & De Mesmaeker, A. (1998) Radical and palladium-mediated cyclizations of ortho-iodo benzyl enamines: Application to solid phase synthesis. Synlett, 1231. #12310

  40. Berteina, S., & De Mesmaeker, A. (1998) Application of radical chemistry to solid support synthesis. Tetrahedron Lett., 39, 5759-5762. #10965

  41. Bertini, V., Lucchesini, F., Pocci, M., & De Munno, A. (1998) 1,3-Dithiane polymers for the supported synthesis of ketones. Tetrahedron Lett., 39, 9263-9266. #12019

  42. Beutel, B.A. (1998) Strategies for screening combinatorial libraries. In E.M. Gordon & J.F.J. Kerwin (Eds.), Combinatorial Chemistry and Molecular Diversity in Drug Discovery. (pp. 421-432). John Wiley & Sons, New York. #11727

  43. Bhalay, G., & Dunstan, A.R. (1998) Facile solid phase synthesis of an activated diazo linker. Tetrahedron Lett., 39, 7803-7806. #11577

  44. Bhalay, G., Cowell, D., Hone, N.D., Scobie, M., & Baxter, A.D. (1998) Multiple solid-phase synthesis of hydantoins and thiohydantoins. Mol. Diversity, 3, 195-198. #11255

  45. Bhandari, A., Jones, D.G., Schullek, J.R., Vo, K., Schunk, C.A., Tamanaha, L.L., Chen, D., Yuan, Z., Needels, M.C., & Gallop, M.A. (1998) Exploring structure-activity relationship around the phosphomannose isomerase inhibitor AF14049 via combinatorial synthesis. Bioorg. Med. Chem. Lett., 8, 2303-2308. #11198

  46. Bianco, A., Zabel, C., Walden, P., & Jung, G. (1998) N-hydroxy-amide analogues of MHC-class I peptide ligands with nanomolar binding affinities. J. Peptide Sci., 4, 471-478. #12313

  47. Bicknell, A.J., Hird, N.W., & Readshaw, S.A. (1998) Efficient robotic synthesis. Multi-component preparation of a tricyclic template by solid phase Tsuge reaction. Tetrahedron Lett., 39, 5869-5872. #10968

  48. Bienayme, H., & Bouzid, K. (1998) Synthesis of rigid hydrophobic tetrazoles using an Ugi multi-component heterocyclic condensation. Tetrahedron Lett., 39, 2735-2738. #10748

  49. Bilodeau, M.T., & Cunningham, A.M. (1998) Solid-supported synthesis of imidazoles: A strategy for direct resin-attachment to the imidazole core. J. Org. Chem., 63, 2800-2801. #10754

  50. Bing, Y. (1998) Monitoring the progress and the yield of solid-phase organic reactions directly on resin supports. Account. Chem. Res., 31, 621-630. #12219

  51. Blackburn, C. (1998) Polymer supports for solid-phase organic synthesis. Biopolymers (Pept. Sci. ), 47, 311-351. #12261

  52. Blackburn, C. (1998) A three-component solid-phase synthesis of 3-aminoimidazol[1,2-a]azines. Tetrahedron Lett., 39, 5469-5472. #10954

  53. Blaskovich, M.A., & Kahn, M. (1998) Polymer-supported acetylide addition to hexa-2,4-dienal. Synthesis-Stuttgart, 965-966. #12236

  54. Blaskovich, M.A., & Kahn, M. (1998) Solid-phase preparation of dienes. J. Org. Chem., 63, 1119-1125. #11798

  55. Bleczinski, C.F., & Richert, C. (1998) Monitoring the hybridization of the components of oligonucleotide mixtures to immobilized DNA via matrix-assisted laser desorption/ionization time-of-flight mass spectrometry. Rapid Commun. Mass Spectrom., 12, 1737-1743. #12315

  56. Bleicher, K.H., & Wareing, J.R. (1998) PhFl polystyrene: A new resin for solid phase organic synthesis. Tetrahedron Lett., 39, 4587-4590. #11171

  57. Bleicher, K.H., & Wareing, J.R. (1998) PhFl acetic acid: A new linker for solid phase organic synthesis. Tetrahedron Lett., 39, 4591-4594. #11164

  58. Blixt, O., & Norberg, T. (1998) Solid-phase enzymatic synthesis of a sialyl Lewis x tetrasaccharide on a sepharose matrix. J. Org. Chem., 63, 2705-2710. #10994

  59. Boeijen, A., Kruijtzer, J.A.W., & Liskamp, R.M.J. (1998) Combinatorial chemistry of hydantoins. Bioorg. Med. Chem. Lett., 8, 2375-2380. #11210

  60. Bogdan, F.M., & Chow, C.S. (1998) The synthesis of allyl- and allyloxycarbonyl-protected RNA phosphoramidites. Useful reagents for solid-phase synthesis of RNAs with base-labile modifications. Tetrahedron Lett., 39, 1897-1900. #10613

  61. Boger, D.L., Goldberg, J., Jiang, W.Q., Chai, W.Y., Ducray, P., Lee, J.K., Ozer, R.S., & Andersson, C.M. (1998) Higher order iminodiacetic acid libraries for probing protein-protein interactions. Bioorg. Med. Chem., 6, 1347-1378. #11825

  62. Bohm, G., Dowden, J., Rice, D.C., Burgess, I., Pilard, J.F., Guilbert, B., Haxton, A., Hunter, R.C., Turner, N.J., & Flitsch, S.L. (1998) A novel linker for the attachment of alcohols to solid supports. Tetrahedron Lett., 39, 3819-3822. #10849

  63. Bondy, S.S. (1998) The role of automation in drug discovery. Curr. Opin. Drug. Disc. Develop., 1, 116-119. #11395

  64. Booth, S., Hermkens, P.H.H., Ottenheijm, H.C.J., & Rees, D.C. (1998) Solid-phase organic reactions III: A review of the literature Nov 96-Dec 97. Tetrahedron, 54, 15385-15443. #12237

  65. Boussie, T.R., Coutard, C., Turner, H., Murphy, V., & Powers, T.S. (1998) Solid-phase synthesis and encoding strategies for olefin polymerization catalyst libraries. Angew. Chem. Int. Ed., 37, 3272-3275. #12139

  66. Boymond, L., Rottlander, M., Cahiez, G., & Knochel, P. (1998) Preparation of highly functionalized Grignard reagents by an iodine-magnesium exchange reaction and its application in solid-phase synthesis. Angew. Chem. Int. Ed., 37, 1701-1703. #11257

  67. Brady, S.F., Stauffer, K.J., Lumma, W.C., Smith, G.M., Ramjit, H.G., Lewis, S.D., Lucas, B.J., Gardell, S.J., Lyle, E.A., Appleby, S.D., Cook, J.J., Holahan, M.A., Stranieri, M.T., Lynch, J.J.Jr., Lin, J.H., Chen, I.W., Vastag, K., Naylor-Olsen, A.M., & Vacca, J.P. (1998) Discovery and development of the novel potent orally active thrombin inhibitor N-(9-hydroxy-9-fluorenecar-boxy)prolyl trans-4-aminocyclohexylmethyl amide (L-372,460): Coapplication of structure-based design and rapid multiple analogue synthesis on solid support. J. Med. Chem., 41, 401-406. #11236

  68. Bray, A.M., Maeji, N.J., Lagniton, L.M., Chiefari, D., James, I.W., Ang, K., Ede, N., Valerio, R.M. & Mason, T.J. (1998) Simultaneous multiple synthesis by the Multipin(TM) method: Techniques for multiple handling,high throughput characterization and reaction optimization on solid phase. In X. Xu, Y. Ye & J.P. Tam (Eds.), Peptides. Biology and Chemistry. Proceedings of the 1996 Chinese Peptide Symposium. (pp. 67. Kluwer/ESCOM, Dordrecht. #14303

  69. Breitenbucher, J.G., Johnson, C.R., Haight, M., & Phelan, J.C. (1998) Generation of a piperazine-2-carboxamide library: A practical application of the phenol-sulfide react and release linker. Tetrahedron Lett., 39, 1295-1298. #10510

  70. Breitenbucher, J.G., & Hui, H.C. (1998) Titanium mediated reductive amination on solid support: Extending the utility of the 4-hydroxy-thiophenol linker. Tetrahedron Lett., 39, 8207-8210. #12009

  71. Brennan, T., Biddison, G., Frauendorf, A., Schwarcz, L., Keen, B., Ecker, D.J., Davis, P.W., Tinder, R., & Swayze, E.E. (1998) Two-dimensional parallel array technology as a new approach to automated combinatorial solid-phase organic synthesis. Biotech. Bioeng. (Comb. Chem. ), 61, 33-45. #10759

  72. Breslow, R. (1998) Bioorganic chemistry: A natural and unnatural science. J. Chem. Educ., 75, 705-718. #10970

  73. Brill, W.K.D., De Mesmaeker, A., & Wendeborn, S. (1998) Solid phase synthesis of levoglucosan derivatives. Synlett, 1085-1090. #12318

  74. Brill, W.K.D., Schmidt, E., & Tommasi, R.A. (1998) Immobilizations of nucleophiles on polystyrene supports. Synlett, 906. #11258

  75. Broddefalk, J., Bergquist, K.E., & Kihlberg, J. (1998) Use of acid-labile protective groups for carbohydrate moieties in synthesis of glycopeptides related to type II collagen. Tetrahedron, 54, 12047-12070. #11828

  76. Brown, D.S., Revill, J.M., & Shute, R.E. (1998) Merrifield, alpha-methoxyphenyl (MAMP) resin: A new versatile solid support for the synthesis of secondary amides. Tetrahedron Lett., 39, 8533-8536. #11946

  77. Brown, R.C.D. (1998) Recent developments in solid-phase organic synthesis. J. Chem. Soc. Perkin Trans. 1, 3293-3320. #11829

  78. Buchardt, J., & Meldal, M. (1998) A chemically inert hydrophilic resin for solid phase organic synthesis. Tetrahedron Lett., 39, 8695-8698. #11962

  79. Buchstaller, H.P. (1998) Solid phase synthesis of oxazolidinones via a novel cyclisation/cleavage reaction. Tetrahedron, 54, 3465-3470. #11050

  80. Bui, C.T., Rasoul, F.A., Ercole, F., Pham, Y., & Maeji, N.J. (1998) Efficiencies of reductive amination reactions on different solid supports. Tetrahedron Lett., 39, 9279-9282. #12020

  81. Bunin, B.A. (1998) The Combinatorial Index. Academic Press, San Diego. ISBN 0121413403 #10496

  82. Burke, T.R., & Zhang, Z.Y. (1998) Protein-tyrosine phosphatases: Structure, mechanism, and inhibitor discovery. Biopolymers, 47, 225-241. #12323

  83. Butenandt, J., Eker, A.P.M., & Carell, T. (1998) Synthesis, crystal structure, and enzymatic evaluation of a DNA-photolesion isostere. Chem. Eur. J., 4, 642-654. #10991

  84. Byk, G., Dubertret, C., Escriou, V., Frederic, M., Jaslin, G., Rangara, R., Pitard, B., Crouzet, J., Wils, P., Schwartz, B., & Scherman, D. (1998) Synthesis, activity, and structure-activity relationship studies of novel cationic lipids for DNA transfer. J. Med. Chem., 41, 224-235. #10751

  85. Byk, G., Soto, J., Mattler, C., Frederic, M., & Scherman, D. (1998) Novel non-viral vectors for gene delivery: Synthesis of a second-generation library of mono-functionalized poly-(guanidinium)amines and their introduction into cationic lipids. Biotechnol. Bioeng., 61, 81-87. #12221

  86. Campian, E., Peterson, M.L., Saneii, H.H., & Furka, A. (1998) Deconvolution by omission libraries. Bioorg. Med. Chem. Lett., 8, 2357-2362. #11207

  87. Cano, M., Camps, F., & Joglar, J. (1998) Solid phase synthesis of cyclopropenes. Tetrahedron Lett., 39, 9819-9822. #12044

  88. Cao, J., Cuny, G.D., & Hauske, J.R. (1998) Ring opening cross-metathesis on solid support: A combinatorial library synthesis of highly functionalized cyclopentanes. Mol. Diversity, 3, 173-179. #10884

  89. Cao, L.Q., Bornscheuer, U.T., & Schmid, R.D. (1998) Lipase-catalyzed solid-phase synthesis of sugar esters. IV. Selectivity of lipases towards primary and secondary hydroxyl groups in carbohydrates. Biocatalysis and Biotransformation, 16, 249-257. #12324

  90. Carroll, C.D., Patel, H., Johnson, T.O., Guo, T., Orlowski, M., He, Z.M., Cavallaro, C.L., Guo, J., Oksman, A., Gluzman, I.Y., Connelly, J., Chelsky, D., Goldberg, D.E., & Dolle, R.E. (1998) Identification of potent inhibitors of Plasmodium falciparum plasmepsin II from an encoded statine combinatorial library. Bioorg. Med. Chem. Lett., 8, 2315-2320. #11200

  91. Casebier, D., & Baldino, C. (1998) Advances in combinatorial chemistry. Innovations in Pharmaceutical Technology, 1, 63-67. #12089

  92. Chaix, C., Minard-Basquin, C., Delair, T., Pichot, C., & Mandrand, B. (1998) Oligonucleotide synthesis on maleic anhydride copolymers covalently bound to silica spherical support and characterization of the obtained conjugates. J. Appl. Polym. Sci., 70, 2487-2497. #12327

  93. Chamoin, S., Houldsworth, S., & Snieckus, V. (1998) The Stille cross coupling reactions on solid support. Link to solution phase directed ortho metalation. An ester linker approach to styryl, biaryl and heterobiaryl carboxylic acids. Tetrahedron Lett., 39, 4175-4178. #10854

  94. Chamoin, S., Houldsworth, S., Kruse, C.G., Bakker, I., & Snieckus, V. (1998) The Suzuki-Miyaura cross coupling reactions on solid support. Link to solution phase directed ortho metalation. The Leznoff acetal linker approach to biaryl and heterobiaryl aldehydes. Tetrahedron Lett., 39, 4179-4182. #10855

  95. Chandrasekhar, S., & Padmaja, M.B. (1998) Practical preparation of first carbon linked polymer bound 1,3-diol. Syn. Commun., 28, 3715-3720. #11834

  96. Chen, C., McDonald, I.A., & Munoz, B. (1998) Synthesis of dihydropyridone scaffolds on solid support: Resin Activation/Capture Approach/REACAP Technology. Tetrahedron Lett., 39, 217-220. #9869

  97. Chen, C., & Munoz, B. (1998) Solid phase synthesis of 2,4-disubstituted pyridine and tetrahydropyridine derivatives: Resin activation/capture approach/REACAP technology. Tetrahedron Lett., 39, 3401-3404. #10805

  98. Chen, C., & Munoz, B. (1998) Solid phase synthesis of N-acyl-2-substituted-dihydro-4-pyridone: Resin activation/capture approach/REACAP technology. Tetrahedron Lett., 39, 6781-6784. #11224

  99. Chen, S., & Janda, K.D. (1998) Total synthesis of naturally occuring prostaglandin F(2alpha) on a non-cross-linked polystyrene support. Tetrahedron Lett., 39, 3943-3946. #10840

  100. Chen, X.T., Sames, D., & Danishefsky, S.J. (1998) Exploration of modalities in building alpha-O-linked systems through glycal assembly: A total synthesis of the mucin-related F1-alpha antigen. J. Amer. Chem. Soc., 120, 7760-7769. #11265

  101. Cheng, J.F., & Mjalli, A.M.M. (1998) Solid-phase synthesis of D2-isoxazolines. Tetrahedron Lett., 39, 939-942. #10488

  102. Chhabra, S.R., Khan, A.N., & Bycroft, B.W. (1998) Versatile Dde-based primary amine linkers for solid phase synthesis. Tetrahedron Lett., 39, 3585-3588. #10809

  103. Chin, J., Fell, B., Pochapsky, S., Shapiro, M.J., & Wareing, J.R. (1998) 2D SECSY NMR for combinatorial chemistry: High-resolution MAS spectra for resin-bound molecules. J. Org. Chem., 63, 1309-1311. #10664

  104. Cho, C.Y., Youngquist, R.S., Paikoff, S.J., Beresini, M.H., Hebert, A.R., Berleau, L.T., Liu, C.W., Wemmer, D.E., Keough, T., & Schultz, P.G. (1998) Synthesis and screening of linear and cyclic oligocarbamate libraries: Discovery of high affinity ligands for GPIIb/IIIa. J. Amer. Chem. Soc., 120, 7706-7718. #11266

  105. Chou, Y.L., Morrissey, M.M., & Mohan, R. (1998) Novel serine-based linker for the solid-phase synthesis of organic compounds. Tetrahedron Lett., 39, 757-760. #10050

  106. Christopher, J., & Lea, L. (1998) Perkin 1 abstracts: Solid phase organic synthesis. J. Chem. Soc. Perkin Trans. 1, vii-x. #11016

  107. Collins, J.L., Blanchard, S.G., Boswell, G.E., Charifson, P.S., Cobb, J.E., Henke, B.R., Hull-Ryde, E.A., Kazmierski, W.M., Lake, D.H., Leesnitzer, L.M., Lehmann, J., Lenhard, J.M., Orband-Miller, L.A., Gray-Nunez, Y., Parks, D.J., Plunkett, K.D., & Tong, W.Q. (1998) N-(2-benzoylphenyl)-L-tyrosine PPAR gamma agonists. 2. Structure-activity relationship and optimization of the phenyl alkyl ether moiety. J. Med. Chem., 41, 5037-5054. #12335

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