Papers on solid phase organic synthesis published in 1994

This list is arranged by the name of the first author. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.

Recently added entries are marked in bold

1. Altava, B., Burguete, M.I., & Luis, S.V. (1994) Functionalization of polystyrene resins with chiral fragments derived from tartaric acid. Tetrahedron, 50, 7535-7542. #1095

2. Anderson, N.G., Anderson, N.L., Taylor, J. & Goodman, J. (1994) Large scale solid phase synthesis. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 371-376). Mayflower Worldwide Limited, Birmingham. #1564

3. Angell, Y.M., Garcia-Echeverria, C., & Rich, D.H. (1994) Comparative studies of the coupling of N-methylated, sterically hindered amino acids during solid-phase synthesis. Tetrahedron Lett., 35, 5981-5984. #5604

4. Arsequell, G., Krippner, L., Dwek, R.A., & Wong, S.Y.C. (1994) Building blocks for solid-phase glycopeptide synthesis: 2-Acetamido-2-deoxy-b-D-glycosides of FmocSerOH and FmocThrOH. J. Chem. Soc. Chem. Commun., 2383-2384. #3025

5. Backes, B.J., & Ellman, J.A. (1994) Carbon-carbon bond-forming methods on solid support. Utilization of Kenner's "Safety-Catch" linker. J. Amer. Chem. Soc., 116, 11171-11172. #2039

6. Bambino, F., Brownlee, R.T.C., & Chiu, F.C.K. (1994) Synthesis of peptides containing a,a dialkyl amino acids. Tetrahedron Lett., 35, 4615-4618. #5898

7. Beattie, K.L. & Hurst, G.D. (1994) Synthesis and use of oligonucleotide libraries. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 69-76). Mayflower Worldwide Limited, Birmingham. #1854

8. Beebe, X., Chiappari, C.L., Kurth, M.J., & Schore, N.E. (1994) Polymer-supported synthesis of cyclic ethers via an intramolecular 1,3-dipolar addition electrophilic cyclization. Abstract. Paper. ACS, 207, 167-167. #1629

9. Borman, S. (1994) Chemical-enzymatic technique used to make carbohydrates, glycopeptides. C&EN, 37-39. #1384

10. Boyd, E.A., Regan, A.C., & James, K. (1994) Synthesis of alkyl phosphinic acids from silyl phosphonites and alkyl halides. Tetrahedron Lett., 35, 4223-4226. #6033

11. Brill, W.K. (1994) Facile methods to recycle nucleosides during solid phase synthesis of oligonucleotides. Tetrahedron Lett., 35, 3041-3044. #14220 NEWOLD

12. Bunin, B.A., & Ellman, J.A. (1994) Increasing the diversity of a 1,4-benzodiazepine library through side-chain functionalization. Polym. Preprint., 35, 983-984. #2163

13. Bunin, B.A., Plunkett, M.J., & Ellman, J.A. (1994) The combinatorial synthesis and chemical and biological evaluation of 1,4-benzodiazepine library. Proc. Natl. Acad. Sci. USA, 91, 4708-4712. #1041

14. Bycroft, B.W., Chan, W.C., Hone, N.D., Millington, S., & Nash, I.A. (1994) Synthesis of the spider toxins nephilatoxin-9 and -11 by a novel solid-phase strategy. J. Amer. Chem. Soc., 116, 7415-7416. #1123

15. Calmes, M., Daunis, J., Hanouneh, A., & Jacquier, R. (1994) Asymmetric supported reactions: Synthesis of chiral amines. Tetrahedron:Asymmetry, 5, 817-820. #1094

16. Campbell, D.A., & Bermak, J.C. (1994) Solid-phase synthesis of peptidylphosphonates. J. Amer. Chem. Soc., 116, 6039-6040. #1086

17. Campian, E., Sebestyen, F. & Furka, A. (1994) Colored and fluorescent solid supports. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 469-472). Mayflower Worldwide Limited, Birmingham. #1871

18. Carell, T., Wintner, E.A., Bashir-Hashemi, A., & Rebek, J.Jr. (1994) A novel procedure for the synthesis of libraries containing small organic molecules. Angew. Chem. Int. Ed., 33, 2059-2061. #2043

19. Carell, T., Wintner, E.A., & Rebek, J.Jr. (1994) A solution-phase screening procedure for the isolation of active compounds from a library of molecules. Angew. Chem. Int. Ed., 33, 2061-2064. #2044

20. Castells, J., Lopez-Calahorra, F., & Yu, Z. (1994) Preparation and reactions of polymer-supported 1- alkoxycarbonylalkylidenearsoranes. An. Quim., 90, 403-406. #3537

21. Chen, C.X., Ahlberg Randall, L.A., Miller, R.B., Jones, A.D., & Kurth, M.J. (1994) "Analogous" organic synthesis of small-compound libraries: Validation of combinatorial chemistry in small-molecule synthesis. J. Amer. Chem. Soc., 116, 2661-2662. #1952

22. Chetverin, A.B., & Kramer, F.R. (1994) Oligonucleotide arrays: New concepts and possibilities. Biotechnology, 12, 1093-1099. #11116

23. Christiansen-Brams, I., Jansson, A.M., Meldal, M., Breddam, K., & Bock, K. (1994) Silyl protection in the solid-phase synthesis of N-linked glycopeptides. Preparation of glycosylated fluorogenic substrates for subtilisins. Bioorg. Med. Chem., 2, 1153-1167. #2302

24. Danishefsky, S.J., Randolph, J.T., Roberge, J.Y., McClure, K.F., & Ruggeri, R.B. (1994) Application of the glycal assembly method in the solid phase: A new strategy for the synthesis of oligosaccharides and glycoconjugates. Polym. Preprint., 35, 977-978. #5626

25. Delatorre, B.G., Avino, A., Tarrason, G., Piulats, J., Albericio, F., & Eritja, R. (1994) Stepwise solid-phase synthesis of oligonucleotide-peptide hybrids. Tetrahedron Lett., 35, 2733-2736. #839

26. Dendrinos, K.G., & Kalivretenos, A.G. (1994) Convenient protection of amines as carbamates using polymer-bound HOBT as catalyst. J. Chem. Soc., 1463-1464. #10971

27. DeOgny, L., Pramanik, B.C., Arndt, L.L., Jones, J.D., Rush, J., Slaughter, C.A., Radolf, J.D., & Norgard, M.V. (1994) Solid-phase synthesis of biologically active lipopeptides as analogs for spirochetal lipoproteins. Peptide Res., 7, 91-97. #849

28. Desai, M.C., Zuckermann, R.N., & Moos, W.H. (1994) Recent advances in the generation of chemical diversity libraries. Drug Develop. Res., 33, 174-188. #1902

29. Deshpande, M.S. (1994) Formation of carbon-carbon bond on solid support: Application of Stille reaction. Tetrahedron Lett., 35, 5613-5614. #1315

30. DeWitt, S.H. (1994) Molecular diversity strategies. Pharmaceut. News, 1, 11-14. #2422

31. DeWitt, S.H., Schroeder, M.C., Stankovic, C.J., Strode, J.E., & Czarnik, A.W. (1994) DIVERSOMER(TM) technology: Solid phase synthesis, automation, and integration for the generation of chemical diversity. Drug Develop. Res., 33, 116-124. #1898

32. Dorman, D., Ceruso, M., & Prestwich, G.D. (1994) Photolytic release of biologically-active molecules from "caged" compounds. Chemtracts:Org. Chem., 7, 322-328. #2120

33. Dumartin, G., Ruel, G., Kharboutli, J., Delmond, B., Connil, M.F., Jousseaume, B., & Pereyre, M. (1994) Straightforward synthesis and reactivity of polymer-supported organotin hydrides. Synlett, 952-954. #2071

34. Epton, R. (1994) Innovation and Perspectives in Solid Phase Synthesis. Mayflower Scientific Limited, Birmingham. ISBN 0951573519 #13447

35. Faja, M., Reese, C.B., Song, Q.L., & Zhang, P.Z. (1994) Facile preparation of acetals and enol ethers derived from 1-arylpiperidin-4-ones. J. Chem. Soc., 191-194. #8394

36. Fitch, W.L., Detre, G., & Holmes, C.P. (1994) High-resolution (1)H NMR in solid-phase organic synthesis. J. Org. Chem., 59, 7955-7956. #2141

37. Frenette, R., & Friesen, R.W. (1994) Biaryl synthesis via Suzuki coupling on a solid support. Tetrahedron Lett., 35, 9177-9180. #2029

38. Ghosh, S., DeWitt, S.H., Mei, H.Y., Sanders, K., & Czarnik, A.W. (1994) Multiple synthesis of cyclic oligonucleotides using diversomer (Tm) technology. Abstract. Paper. ACS, 208, 240-240. #774

39. Gilchrist, T.L. (1994) Synthesis of aromatic heterocycles [review]. J. Chem. Soc., 615-628. #10676

40. Goodwin, J.T., Stanick, W.A., & Glick, G.D. (1994) Improved solid-phase synthesis of long oligoribonucleotides: Application to tRNA(phe) and tRNA(gly). J. Org. Chem., 59, 7941-7943. #2142

41. Gordon, E.M., Barrett, R.W., Dower, W.J., Fodor, S.P.A., & Gallop, M.A. (1994) Applications of combinatorial technologies to drug discovery. 2. Combinatorial organic synthesis, library screening strategies, and future directions. J. Med. Chem., 37, 1385-1401. #1001

42. Green, M., McGeehan, G.M., Anderegg, R.S., Bickett, D.M., Kassel, D., Aquino, C.J., Sugg, E.E., Millington, S., Norwod, D.L., Wiseman, J.S. & Bermann, J. (1994) Protease substrate mapping. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 239-244). Mayflower Worldwide Limited, Birmingham. #1860

43. Green, O.M. (1994) A rapid dealkylation of phosphonate diester for the preparation of 4-phosphonomethylphenylalanine-containing peptides. Tetrahedron Lett., 35, 8081-8084. #6556

44. Hagrman, D., Zubieta, C., Rose, D.J., Zubieta, J., & Haushalter, R.C. (1994) Composite solids constructed from one-dimensional coordination polymer matrices and molybdenum oxide subunits - polyoxomolybdate clusters within [(cu(4,4'-bpy))(4)mo8o26] and [(ni(h2o)(2)(4,4'- bpy)(2))(2)mo8o26] and one-dimensional oxide chains in [(cu(4,4'- bpy))(4)mo15o47]center-dot-8h(2)o. Angew. Chem., 873-876. #9099

45. Halcomb, R.L., Huang, H., & Wong, C.H. (1994) Solution- and solid-phase synthesis of inhibitors of H. pylori attachment and E-selectin-mediated leukocyte adhesion. J. Amer. Chem. Soc., 116, 11315-11322. #2118

46. Hebert, N., Davis, P.W., DeBaets, E.L., & Acevedo, O.L. (1994) Synthesis of N-substituted hydroxyprolinol phosphoramidites for the preparation of combinatorial libraries. Tetrahedron Lett., 35, 9509-9512. #2078

47. Hong, F., Zaidi, J., Pang, Y.P., Cusack, B., & Richelson, E. (1994) Design, synthesis and pharmacological evaluation of active pyrrole based, nonpeptidic analogues of neurotensin(8-13). J. Chem. Soc., 2997-3003. #10218

48. Hovinen, J., Guzaev, A., Azhayev, A., & Lonnberg, H. (1994) Novel solid supports for the preparation of 3'-derivatized oligonucleotides: Introduction of 3'-alkylphosphate tether groups bearing amino, carboxy, carboxamido and mercapto functionalities. Tetrahedron, 50, 7203-7218. #8550

49. Hutchins, S.M., & Chapman, K.T. (1994) A general method for the solid phase synthesis of ureas. Tetrahedron Lett., 35, 4055-4058. #1098

50. Jansson, A.M., Meldal, M. & Bock, K. (1994) N-Fmoc-8-amino-2,8-dideoxy-b-KDO pentafluorophenyl ester used as a building block in multiple column solid phase neoglycopeptide synthesis. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 559-562). Mayflower Worldwide Limited, Birmingham. #1875

51. Kates, S.A., de la Torre, B.G., Eritja, R., & Albericio, F. (1994) Solid-phase N-glycopeptide synthesis using allyl side-chain protected Fmoc-amino acids. Tetrahedron Lett., 35, 1033-1034. #3822

52. Kim, M.H., & Patel, D.V. (1994) "BOP" as a reagent for mild and efficient preparation of esters. Tetrahedron Lett., 35, 5603-5606. #3675

53. Koepper, S. (1994) Polymer-supported enzymic synthesis on a preparative scale. Carbohyd. Res., 265, 161-166. #2608

54. Kopper, S., & Zehavi, U. (1994) Improved acceptor polymers for enzymic glycosylation. React. Polym., 22, 171-180. #5288

55. Krchnak, V., Cabel, D., Weichsel, A., & Flegelova, Z. (1994) Esterification of polymer-supported hydroxyl groups using the Mitsunobu reaction. Lett. Peptide Sci., 1, 277-282. #2427

56. Kundu, B., Tripathi, M., & Shukla, S. (1994) Solid phase synthesis of muramyl dipeptide and its analogues. Ind. J. Chem. B-Org. Chem. Med. Chem., 33B, 1180-1182. #2602

57. Kuper, J., Conrad, O., & Krebs, B. (1994) Selenoboratoborates [b-12(bse3)(6)](8-): A new class of chalcogen-substituted icosahedral boron clusters. Angew. Chem., 1903-1904. #10257

58. Kurth, M.J., Randall, L.A.A., Chen, C., Melander, C., Miller, R.B., McAlister, K., Reitz, G., Kang, R., Nakatsu, T., & Green, C. (1994) Library-based lead compound discovery: Antioxydants by an analogous synthesis deconvolutive assay strategy. J. Org. Chem., 59, 5862-5864. #1635

59. Le Bec, C., & Wickstrom, E. (1994) Stereospecific Grignard activated coupling of a deoxynucleoside methylphosphonate on a polyethylene glycol support. Tetrahedron Lett., 35, 9525-9528. #2085

60. Lebl, M., Krchnak, V., Sepetov, N.F., Nikolaev, V., Stierandova, A., Safar, P., Seligmann, B., Strop, P., Thorpe, D., Felder, S., Lake, D.F., Lam, K.S. & Salmon, S.E. (1994) One bead-one structure libraries. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 233-238). Mayflower Worldwide Limited, Birmingham. #512

61. Lebl, M., Krchnak, V., Safar, P., Stierandova, A., Sepetov, N.F., Kocis, P. & Lam, K.S. (1994) Construction and screening of libraries of peptide and non- peptide structures. In J.W. Crabb (Ed.), Techniques in Protein Chemistry V. (pp. 541-548). Academic Press, San Diego. #510

62. Lebl, M., Krchnak, V., Stierandova, A., Safar, P., Kocis, P., Nikolaev, V., Sepetov, N.F., Ferguson, R., Seligmann, B., Lam, K.S. & Salmon, S.E. (1994) Nonsequenceable and/or nonpeptide libraries. In R.S. Hodges & J.A. Smith (Eds.), Peptides: Chemistry, Structure and Biology,Proc.13.APS. (pp. 1007-1008). ESCOM, Leiden. #513

63. Liao, W.S., & Lu, D.P. (1994) Progress on solid-phase syntheses of oligosaccharides [in Chinese]. Youji Huaxue, 14, 571-580. #2697

64. Liskamp, R.M.J. (1994) Opportunities for new chemical libraries. Unnatural biopolymers and diversomers. Angew. Chem. Int. Ed., 33, 633-636. #932

65. Look, G.C., Holmes, C.P., Chinn, J.P., & Gallop, M.A. (1994) Methods for combinatorial organic synthesis: The use of fast 13C NMR analysis for gel phase reaction monitoring. J. Org. Chem., 59, 7588-7590. #2106

66. Lowe, G., & Vilaivan, T. (1994) Solid-phase synthesis of novel peptide nucleic acids. J. Chem. Soc., 555-560. #9173

67. Markiewicz, W.T., Adrych-Rozek, K., Markiewicz, M., Zebrowska, A. & Astriab, A. (1994) Synthesis of oligonucleotides permanently linked with solid supports for use as synthetic oligonucleotide combinatorial libraries. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 339-346). Mayflower Worldwide Limited, Birmingham. #1866

68. Mathieux, N., Paulsen, H., Meldal, M., & Bock, K. (1994) Synthesis of glycopeptide sequences of repeating units of the mucins MUC 2 and MUC 3 containing oligosaccharide side-chains with core 1, core 2, core 3, core 4 and core 6 structure. J. Chem. Soc., 2359-2368. #10283

69. Medzihradszky, D., Chen, S.L., Kenyon, G.L., & Gibson, B.W. (1994) Solid-phase synthesis of adenosine phosphopeptides as potential bisubstrate inhibitors of protein kinases. J. Amer. Chem. Soc., 116, 9413-9419. #1670

70. Mehta, S., Meldal, M., Ferro, V., Duus, J.O., & Bock, K. (1994) Internally quenched fluorogenic, alpha-helical dimeric peptides and glycopeptides for the evaluation of the effect of glycosylation on the conformation of peptides. J. Chem. Soc., 1365-1374. #9104

71. Meldal, M. (1994) Multiple column synthesis of quenched solid-phase bound fluorogenic substrates for characterization of endoprotease specificity. Methods: A Companion to Methods in Enzymology, 6, 417-424. #993

72. Meldal, M. (1994) Recent development in glycopeptide and oligosaccharide synthesis. Curr. Opin. Struct. Biol., 4, 710-718. #4910

73. Menicagli, R., Malanga, C., & Peluso, P. (1994) Selective mono- or dialkoxylation of 2,4,6-trichloro-1,3,5-triazine in solid-liquid phase transfer conditions. Syn. Commun., 24, 2153-2158. #1099

74. Mereyala, H.B., Gurrala, S.R., & Gadikota, R.R. (1994) Stereoselective synthesis of alpha-O-fucosylated serine, threonine, tyrosine and saccharides. J. Chem. Soc., 3179-3182. #10291

75. Miller, S.M., Simon, R.J., Ng, S., Zuckermann, R.N., Kerr, J.M., & Moos, W.H. (1994) Proteolytic studies of homologous peptide and N-substituted glycine peptoid oligomers. Bioorg. Med. Chem. Lett., 4, 2657-2662. #2316

76. Montserrat, F.X., Grandas, A., Eritja, R., & Pendroso, E. (1994) Criteria for the economic large scale solid-phase synthesis of oligonucleotides. Tetrahedron, 50, 2617-2622. #3980

77. Moon, H.S., Schore, N.E., & Kurth, M.J. (1994) A polymer-supported C2-symmetric chiral auxiliary: Preparation of non-racemic 3,5-disubstituted-gamma-butyrolactones. Tetrahedron Lett., 35, 8915-8918. #2041

78. Nestler, H.P., Bartlett, P.A., & Still, W.C. (1994) A general method for molecular tagging of encoded combinatorial chemistry libraries. J. Org. Chem., 59, 4723-4724. #1312

79. Norberg, T., Luning, B., & Tejbrant, J. (1994) Solid-phase synthesis of O-glycopeptides. Methods Enzymol., 247, 87-106. #2606

80. Ostresh, J.M., Husar, G.M., Blondelle, S.E., Dorner, B., Weber, P.A., & Houghten, R.A. (1994) "Libraries from libraries": Chemical transformation of combinatorial libraries to extend the range and repertoire of chemical diversity. Proc. Natl. Acad. Sci. USA, 91, 11138-11142. #1921

81. Pascal, R., Chauvey, D., & Sola, R. (1994) Carbonyl-protecting groups convertible into activating groups.Carbamates of o-aminoanilides are precursors of reactive N-acylureas. Tetrahedron Lett., 35, 6291-6294. #275

82. Patek, M. & Lebl, M. (1994) "Safety-Catch" anchoring linkages and protecting groups in solid-phase peptide synthesis. In R.S. Hodges & J.A. Smith (Eds.), Peptides: Chemistry, Structure and Biology,Proc.13.APS. (pp. 146-148). ESCOM, Leiden. #1004

83. Patek, M., Drake, B., & Lebl, M. (1994) All-cis cyclopentane scaffolding for combinatorial solid phase synthesis of small non-peptide compounds. Tetrahedron Lett., 35, 9169-9172. #1346

84. Paulsen, H., Bielfeldt, T., Peters, S., Meldal, M., & Bock, K. (1994) A new strategy for the solid-phase synthesis of O-glycopeptides via 2-azido-glycopeptides. Liebigs Ann. Chem., 369-379. #3981

85. Pei, Y., & Moos, W.H. (1994) Post-modification of peptoid side chains: [3+2] Cycloaddition of nitrile oxides with alkenes and alkynes on the solid-phase. Tetrahedron Lett., 35, 5825-5828. #11601

86. Pei, Y.H., & Moos, W.H. (1994) Post-modification of peptoid side chains: [3+2] cycloaddition of nitrile oxides with alkenes and alkynes on the solid-phase. Tetrahedron Lett., 35, 5825-5828. #217

87. Ramaraj, B., & Radhakrisnan, G. (1994) Modification of the dynamic swelling behaviour of poly(2-hydroxyethyl methacrylate)hydrogels in water through interpenetrating polymer networks (IPNs). Polymer, 35, 2167-2173. #1081

88. Rao, M.V., & MacFarlane, K. (1994) Solid phase synthesis of phosphorothioate oligonucleotides using benzytriethylammonium tetrathiomolybdate as a rapid sulfur transfer reagent. Tetrahedron Lett., 35, 6741-6744. #14221 NEWOLD

89. Ravindranathan, T., Chavan, S.P., & Awachat, M.M. (1994) Polymer supported nitrobenzaldehyde: Efficient, highly selective catalytic, deprotection of oxathioacetals. Tetrahedron Lett., 35, 8835-8838. #5676

90. Reddy, M.P., Michael, M.A., Farooqui, F., & Girgis, N.S. (1994) New and efficient solid support for the synthesis of nucleic acids. Tetrahedron Lett., 35, 5771-5774. #2562

91. Richter, L.S., & Gadek, T.R. (1994) A surprising observation about Mitsunobu reactions in solid phase synthesis. Tetrahedron Lett., 35, 4705-4706. #1097

92. Robles, J., Pedroso, E., & Grandas, A. (1994) Stepwise solid-phase synthesis of the nucleopeptide Phac-Phe-Val- Ser(p3'ACT)-Gly-OH. J. Org. Chem., 59, 2482-2486. #575

93. Rose, K. (1994) Artificial proteins made by parallel assembly. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 21-28). Mayflower Worldwide Limited, Birmingham. #1853

94. Rothe, M., & Zieger, M. (1994) Polymer-supported synthesis of series of macrocyclic oligoesters. Tetrahedron Lett., 35, 9011-9012. #2053

95. Rozners, E., Westman, E., & Stromberg, R. (1994) Evaluation of 2'-hydroxyl protection in RNA-synthesis using the H-phosphonate approach. Nucl. Acid. Res., 22, 94-99. #7593

96. Saha, U.K., & Schmidt, R.R. (1994) Efficient synthesis of O-(2-acetamido-2-deoxy-beta-D-glucopyranosyl)-serine and -threonine building blocks for glycopeptide formation. J. Chem. Soc., 1855-1860. #9485

97. Schuster, M., Wang, P., Paulson, J.C., Wong, C.H., Kanie, O., & Ogawa, T. (1994) Solid-phase chemical-enzymatic synthesis of glycopeptides and oligosaccharides. Chemtracts:Org. Chem., 7, 196-198. #1934

98. Schuster, M., Wang, P., Paulson, J.C., & Wong, C.H. (1994) Solid-phase chemical-enzymatic synthesis of glycopeptides and oligosaccharides. J. Amer. Chem. Soc., 116, 1135-1136. #998

99. Scremin, C.L., Zhou, L., Srinivassachar, K., & Beaucage, S. (1994) Stepwise regeneration and recovery of deoxyribonucleoside phosphoramidite monomers during solid-phase oligonucleotide synthesis. J. Org. Chem., 59, 1963-1966. #14219 NEWOLD

100. Setty-Fichman, M., Blum, J., Sasson, Y., & Eisen, M. (1994) Polystyrene-supported RhCl3-quarternary ammonium ion pair as a long-lived, efficient and recyclabe catalyst. Tetrahedron Lett., 35, 781-784. #5687

101. Shapiro, G., & Buechler, D. (1994) Mild and rapid azide-mediated, palladium catalyzed cleavage of allylester based protecting groups. Tetrahedron Lett., 35, 5421-5424. #5688

102. Simon, R.J., Martin, E.J., Miller, S.M., Zuckermann, R.N., Blaney, J.M. & Moos, W.H. (1994) Using peptoid libraries [oligo N-substituted glycines] for drug discovery. In J.W. Crabb (Ed.), Techniques in Protein Chemistry V. (pp. 533-539). Academic Press, San Diego. #1038

103. Southern, E.M., Case-Green, S.C., Elder, J.K., Johnson, M., Mir, K.U., Wang, L., & et al. (1994) Arrays of complementary oligonucleotides for analysing the hybridisation behaviour of nucleic acids. Nucl. Acid. Res., 22, 1368-1373. #11129

104. Spetzler, J.C., Meldal, M., Felding, J., Vedso, P., & Begtrup, M. (1994) Novel acylation catalysts in peptide synthesis: Derivatives of N-hydroxytriazoles and N-hydroxytetrazoles. J. Chem. Soc., 1727-1732. #10947

105. Stankova, M., Issakova, O., Sepetov, N.F., Krchnak, V., Lam, K.S., & Lebl, M. (1994) Application of one-bead one-structure approach to identification of nonpeptidic ligands. Drug Develop. Res., 33, 146-156. #1008

106. Stankovic, C.J., DeWitt, S.H., Schroeder, M.C., Kiely, J.S., Cody, D.M.R. & Pavia, M.R. (1994) Diversomer libraries a novel approach to chemical diversity. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 391-396). Mayflower Worldwide Limited, Birmingham. #1869

107. Story, S.C., & Aldrich, J.V. (1994) Side-product formation during cyclization with HBTU on a solid support. Int. J. Peptide Prot. Res., 43, 292-296. #1451

108. Sucholeiki, I. (1994) Solid-phase photochemical C-S bond cleavage of thioethers. A new approach to the solid-phase production of non-peptide molecules. Tetrahedron Lett., 35, 7307-7310. #2102

109. Sugawara, T., Kato, S., & Okamoto, S. (1994) Development of fully automated synthesis systems. J. Automation Chem., 16, 33. #8295

110. Thompson, L.A., & Ellman, J.A. (1994) Straightforward and general method for coupling alcohols to solid supports. Tetrahedron Lett., 35, 9333-9336. #2112

111. Truffert, J.C., Lorthioir, O., Asseline, U., Thuong, N.T., & Brack, A. (1994) On-line solid phase synthesis of oligonucleotide-peptide hybrids using silica supports. Tetrahedron Lett., 35, 2353-2356. #2686

112. Varadi, G., Toth, G.K., & Penke, B. (1994) A new synthesis of Rink's polymer, 4-(2',4'-dimethoxyphenylhydroxymethyl)phenoxymethylpolystyrene. Int. J. Peptide Prot. Res., 43, 29-30. #7940

113. Virgilio, A.A., & Ellman, J.A. (1994) Simultaneous solid-phase synthesis of b-turn mimetics incorporating side-chain functionality. J. Amer. Chem. Soc., 116, 11580-11581. #2117

114. Wakamiya, T., Saruta, K., Yasuoka, J., & Kusumoto, S. (1994) An efficient procedure for solid-phase synthesis of phosphopeptides by the Fmoc strategy. Chem. Lett., 1099-1102. #2559

115. Yan, L., Taylor, C.M., Goodnow, R.J., & Kahne, D. (1994) Glycosylation on the Merrifield resin using anomeric sulfoxides. J. Amer. Chem. Soc., 116, 6953-6954. #1115

116. Young, J.K., Nelson, J.C., & Moore, J.S. (1994) Synthesis of sequence specific phenylacetylene oligomers on an insoluble solid support. J. Amer. Chem. Soc., 116, 10841-10842. #2037

117. Yu, K.L., Deshpande, M.S., & Vyas, D.M. (1994) Heck reactions in solid phase synthesis. Tetrahedron Lett., 35, 8919-8922. #1308

118. Zambias, R.A., Boulton, D.A., & Griffin, P.R. (1994) Microchemical structural determination of a peptoid covalently bound to a polymeric bead by matrix-assisted laser desorption ionization time-of-flight mass spectrometry. Tetrahedron Lett., 35, 4283-4286. #1096

119. Zhao, Z., & Felix, A.M. (1994) Solid-phase synthesis of extended lactam ring systems: Preparation of amino acid a-fluorenylmethyl esters for the synthesis of reverse-extended lactams. Peptide Res., 7, 218-223. #1120

120. Zuckermann, R.N., & Goff, D.A. (1994) Synthesis of (N-substituted)-glycine polymers of defined length and sequence. Polym. Preprint., 35, 975-976. #5734

121. Zuckermann, R.N., Figliozzi, G.M., Banville, S.C., Kerr, J.M., Siani, M.A., Martin, E.J., Brown, E.G. & Wang, L. (1994) Automated tools for the production of non-natural molecular diversity. In R. Epton (Ed.), Innovation and Perspectives in Solid Phase Synthesis. (pp. 397-402). Mayflower Worldwide Limited, Birmingham. #1870

122. Zuckermann, R.N., Martin, E.J., Spellmeyer, D.C., Stauber, G.B., Shoemaker, K.R., Kerr, J.M., Figliozzi, G.M., Goff, D.A., Siani, M.A., Simon, R.J., Banville, S.C., Brown, E.G., Wang, L., Richter, L.S., & Moos, W.H. (1994) Discovery of nanomolar ligands for 7-transmembrane G-protein-coupled receptors from a diverse N-(substituted)glycine peptoid library. J. Med. Chem., 37, 2678-2685. #1171