Papers on solid phase organic synthesis published in 1993

This list is arranged by the name of the first author. Any omissions, mistakes and inconsistencies please communicate to the authors of compilation (michal@5z.com). (If you are pointing to any reference, please use its ID# -- the last number in the reference.) You are welcome to use this compilation in your work. Proper way to quote it in your paper is: Lebl M., Leblova Z.: Dynamic database of references in molecular diversity. Internet http://www.5z.com.

Recently added entries are marked in bold

1. Andrews, D.M., & Seale, P.W. (1993) Solid-phase synthesis of O-mannosylated peptides: Two strategies compared. Int. J. Peptide Prot. Res., 42, 165-170. #5845

2. Berg, R.H., Nielsen, P.E., Buchardt, O. & Egholm, M. (1993) Peptide nucleic acids (PNA): A new strategy toward the rational design of DNA mimics. In C.H. Schneider & A.N. Eberle (Eds.), Peptides 1992, Proc.22.EPS. (pp. 152-153). ESCOM, Leiden. #4530

3. Burdick, D.J., Struble, M.E., & Burnier, J.P. (1993) Solid phase synthesis of peptide para-nitroanilides. Tetrahedron Lett., 34, 2589-2592. #277

4. Chen, Z.P., & Hemmasi, B. (1993) Synthesis of phytochelatins by the continuous flow solid phase procedure. Biol. Chem. Hoppe-Seyler, 374, 1057-1062. #6168

5. Chiu, H.C., Zalipsky, S., Kopeckova, P., & Kopecek, J. (1993) Enzymatic activity of chymotrypsin and its poly(ethylene glycol) conjugates toward low and high molecular weight substrates. Bioconjug. Chem., 4, 290-295. #1377

6. Cho, C.Y., Moran, E.J., Cherry, S.R., Stephans, J.C., Fodor, S.P.A., Adams, C.L., Sundaram, A., Jacobs, J.W., & Schultz, P.G. (1993) An unnatural biopolymer. Science, 261, 1303-1305. #478

7. Chorev, M., & Goodman, M. (1993) A dozen years of retro-inverso peptidomimetics. Account. Chem. Res., 26, 266-273. #4526

8. Christensen, M.K., Meldal, M., & Bock, K. (1993) Synthesis of mannose 6-phosphate-containing disaccharide threonine building blocks and their use in solid-phase glycopeptide synthesis. J. Chem. Soc. Perkin Trans. 1, 1453-1460. #1298

9. Christiansen-Brams, I., Meldal, M., & Bock, K. (1993) Silyl protection in the solid-phase synthesis of N-linked neoglycopeptides. One-step deprotection of fully protected neoglycopeptides. Tetrahedron Lett., 34, 3315-3318. #1302

10. Danishefsky, S.J., McCure, K.F., Randolph, J.T., & Ruggeri, R.B. (1993) A strategy for the solid-phase synthesis of oligosaccharides. Science, 260, 1307-1309. #2371

11. DeWitt, S.H., Kiely, J.S., Stankovic, C.J., Schroeder, M.C., Cody, D.M.R., & Pavia, M.R. (1993) DIVERSOMERS: An approach to nonpeptide nonoligomeric chemical diversity. Derwent Drug File, 30, 45727-45728. #2418

12. DeWitt, S.H., Stankovic, C.J. & Schroeder, M.C. (1993) The DIVERSOMER approach: Integration and automation of multiple, simultaneous solid phase synthesis. In J.R. Stimatitis & G.L. Hawk (Eds.), Advances in Laboratory Automation-Robotics. (pp. 248-263). Zymark Corporation, Hopkinton,MA. #2373

13. DeWitt, S.H., Kiely, J.S., Stankovic, C.J., Schroeder, M.C., Cody, D.M.R., & Pavia, M.R. (1993) "Diversomers": An approach to nonpeptide, nonoligomeric chemical diversity. Proc. Natl. Acad. Sci. USA, 90, 6909-6913. #2372

14. Ecker, D.J., Vickers, T.A., Hanecak, R., Driver, V., & Anderson, K. (1993) Rational screening of oligonucleotide combinatorial libraries for drug discovery. Nucl. Acid. Res., 21, 1853-1856. #668

15. Jensen, K.J., Meldal, M., & Bock, K. (1993) Glycosylation of phenols: Preparation of 1,2-cis and 1,2-trans glycosylated tyrosine derivatives to be used in solid-phase glycopeptide synthesis. J. Chem. Soc. Perkin Trans. 1, 2119-2129. #1300

16. Kaljuste, K., & Und n, A. (1993) New method for the synthesis of N-methyl amino acids containing peptides by reductive methylation of amino groups on the solid phase. Int. J. Peptide Prot. Res., 42, 118-124. #1172

17. Leznoff, C.C., McArthur, C.R., & Qin, Y. (1993) Phthalocyanine-modified silica gels and their application in the purification of unsymmetrical phthalocyanines. Can. J. Chem., 71, 1319-1326. #2457

18. Lopez, E., Chypre, C., Alpha, B., & Mathis, G. (1993) Europium (III) trisbipyridine cryptate label for time-resolved fluorescence detection of PCR products fixed on a solid support. Clin. Chem., 39, 196-201. #9967

19. Maskos, U., & Southern, E.M. (1993) A study of oligonucleotide reassociation using large arrays of oligonucleotides synthesized on a glass support. Nucl. Acid. Res., 21, 4663-4669. #10571

20. Mergler, M. and Nyfeler, R. Polymeric diphenyldiazomethane: A useful resin for SPPS and solid phase organic synthesis. 1993. #12541

21. Moos, W.H., Green, G.D., & Pavia, M.R. (1993) Recent advances in the generation of molecular diversity. Annu. Rep. Med. Chem., 28, 315-324. #701

22. Nikolaiev, V., Stierandova, A., Krchnak, V., Seligmann, B., Lam, K.S., Salmon, S.E., & Lebl, M. (1993) Peptide-encoding for structure determination of nonsequenceable polymers within libraries synthesized and tested on solid-phase supports. Peptide Res., 6, 161-170. #509

23. Pulley, S.R., & Hegedus, L.S. (1993) Solid-phase, solution, and segment condensation peptide syntheses incorporating chromium carbene complex-derived nonproteinogenic ("unnatural") amino acid fragments. J. Amer. Chem. Soc., 115, 9037-9047. #1448

24. Saha, A.K., Sardaro, M., Waychunas, C., Delecki, D., Kutny, R., Cavanaugh, P., Yawman, A., Upson, D.A., & Kruse, L.I. (1993) Diisopropylsilyl-linked oligonucleotide analogs: Solid-phase synthesis and physicochemical properties. J. Org. Chem., 58, 7827-7831. #5685

25. Schwabacher, A.W., & Maynard, T.L. (1993) Preparation of peptide thioacids using the Kaiser oxime resin. Tetrahedron Lett., 34, 1269-1270. #2459

26. Shepard, R.C. (1993) Solid-phase synthesis. Trends Biotech., 11, 492-493. #11654

27. Smigol, V., & Svec, F. (1993) Preparation and properties of uniform beads based on macroporous glycidyl methacrylate-ethylene dimethacrylate copolymer: Use of chain transfer agent for control of the pore-size distribution. J. Appl. Polym. Sci., 48, 2033-2039. #634

28. Smigol, V., Svec, F., & Frechet, J.M.J. (1993) Use of polymeric catalysts in the pore-size-specific functionalization of porous polymers. Macromolecules, 26, 5615-5620. #645

29. Tamamura, H., Nakamura, J., Noguchi, K., Funakoshi, S., & Fujii, N. (1993) Acceleration of the N(alpha)-deprotection rate by the addition of m-cresol to diluted methanesulfonic acid and its application to the Z(OMe)-based solid-phase syntheses of human pancreastatin-29 and magainin-1. Chem. Pharm. Bull. Tokyo, 41, 954-957. #7837

30. Tian, Z., Gu, C., Roeske, R.W., Zhou, M., & Van Etten, R.L. (1993) Synthesis of phosphotyrosine-containing peptides by the solid-phase method. A re-examination of the use of Boc-Tyr(PO3Bzl2)-OH. Int. J. Peptide Prot. Res., 42, 155-158. #7861

31. Tourwe, D., Piron, J., Defreyn, P., & Van Binst, G. (1993) A new method for the solid phase synthesis of hydroxyethylamine peptide bond isosteres. Synthesis of an HIV-1 protease inhibitor and of a beta-casomorphin-5 analogue. Tetrahedron Lett., 34, 5499-5502. #7873

32. Wenschuh, H., Beyermann, M., Krause, E., Carpino, L.A., & Bienert, M. (1993) Efficient solid phase assembly of peptides bearing contiguous highly hindered Aib residues via Fmoc Aib fluoride. Tetrahedron Lett., 34, 3733-3736. #8008

33. Wright, P., Lloyd, D., Rapp, W., & Andrus, A. (1993) Large scale synthesis of oligonucleotides via phosphoramidite nucleosides and a high-loaded polystyrene support. Tetrahedron Lett., 34, 3373-3376. #3095

34. Zhou, Y., & Romano, L.J. (1993) Solid-phase synthesis of oligonucleotides containing site- specific N-(2'-deoxyguanosin-8-yl)-2-(acetylamino)fluorene adducts using 9-fluorenylmethoxycarbonyl as the base-protecting group. Biochemistry, 32, 14043-14052. #706