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PAPERS PUBLISHED
- Makarov, M.; Sanchez Rocha, A.C.; Krystufek, R.; Cherepashuk, I.; Dzmitruk, V.;
Charnavets, T.; Faustino, A.M; Lebl, M.; Fujishima, K.; Fried, S.D.; Hlouchova, K. Early selection of the amino acid alphabet was adaptively shaped by biophysical constraints of foldability . J.Am.Chem.Soc. 2023, 145, 5320–5329. 2023JACS_5320.pdf
- Lebl, M. How to make sure that you will get the Nobel Prize . Chem. Listy 2023, 117 , 485–486. 2023ChemListy.pdf
- Pazderkova, M.; Bednarova, L.; Dlouha, H.; Lebl, M.; Hlavacek, J.; Setnicka, V.; Urbanova, M.; Hynie, S.; Klenerova, V.; Baumruk, V.; Malon, P.. Electronic and vibrational optical activity of several peptides related to neurohypophyseal hormones: Disulfide group conformation. Biopolymers 2012, 97 , 923–932. 2012Biopolymers.pdf
- Lebl-Rinnova, M.; Tran, H. N.; Lebl, M. Modified synthesis of safety catch acid-labile (SCAL) linker. In: Peptides, Building Bridges: The Proceedings of The Twenty-Second American Peptide Symposium, Lebl, M., Ed.; Prompt Scientific Publishing: San Diego, 2011; pp 40-41. 2011Proc22APS_40.pdf
- Lebl, M.; Heiner, D.; Jones, A. C.; Fambro, S. P.; Nibbe, M. J.; Burgett, S. R.; Ellman, B. M. Automatic oligonucleotide synthesizer utilizing the concept of parallel processing. Collection Symposium Series 2011, 12, 264-267. 2011CCCC.pdf
- Lebl, M.; Slaninova, J. Ala-Walk analogs of oxytocin - HPLC-based conformational studies. In: Peptides, Building Bridges: The Proceedings of The Twenty-Second American Peptide Symposium, Lebl, M., Ed.; Prompt Scientific Publishing: San Diego, 2011; pp 316-317. 2011Proc22APS_316.pdf
- Lebl, M. Combinatorial/Library Peptide Synthesis. In: Amino Acids, Peptides and Proteins in Organic Chemistry, Hughes, A. B., Ed.; Wiley: Weinheim, 2011; pp 395-449. 2011AAPeptProt.pdf
- Schroeder, M. A.; Salloum, K. S.; Perbost, M.; Lebl, M.; Posner, J. D. Radial flow electroosmotic pump. Sensor. Actuator. A-Phys. 2011, 169 (1), 250-255. 2011SensorsActuators.pdf
- Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Srinivasan, A.; Shults, M. D.; Zhao, C.; Musmacker, J.; Nelson, N.; Barker, D. L.; Lebl, M. A high-complexity, multiplexed solution-phase assay for profiling protease activity on microarrays. Comb. Chem. High Throughput Screening 2008, 11, 24-35. 2008CombChemHighThrScr.pdf
- Remacle, A. G.; Shiryaev, S. A.; Oh, E. S.; Cieplak, P.; Srinivasan, A.; Wei, G.; Liddington, R. C.; Ratnikov, B. I.; Parent, A.; Desjardins, R.; Day, R.; Smith, J. W.; Lebl, M.; Strongin, A. Y. Substrate cleavage analysis of furin and related proprotein convertases. Journal of Biological Chemistry 2008, 283 (30), 20897-20906. 2008JBiolChem.pdf
- Kermani, B. G.; Kozlov, I. A.; Melnyk, P. C.; Zhao, C.; Hachmann, J. P.; Lebl, M. Using support vector machine regression to model the retention of peptides in immobilized metal-affinity chromatography. Sensors. and Actuators B: Chemical 2007, 125, 149-157. 2007SensActBChem.pdf
- Kozlov, I. A.; Kermani, B. G.; Melnyk, P. C.; Barker, D. L.; Zhao, C.; Hachmann, J. P.; Lebl, M. Study of the retention of histidine containing peptides on nickel column. J. Chromatogr. Sci. 2007, 45, 207-211. span style="text-decoration: underline;">2007JChromSci.pdf
- Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Barker, D. L.; Lebl, M.; Zhao, C. Evaluation of different chemical strategies for conjugation of oligonucleotides to peptides. Nucleosides, Nucleotides & Nucleic Acids 2007, 26 (10), 1353-1357. 2007NuclNuclNuclAcids.pdf
- Lebl, M.; Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Srinivasan, A.; Shults, M. D.; Musmacker, J.; Nelson, N.; Kermani, B. G.; Zhao, C.; Barker, D. L. High complexity protease and kinase profiling solution assays with readout on randomly assembled microarrays. In: Proc.29th Eur. Pept. Symp., Gdansk, 2006, 2007; p in press. 2007Proc29EPS.pdf
- Lebl, M.; Pistek, C.; Hachmann, J. P.; Mudra, P.; Pesek, V.; Pokorny, V.; Poncar, P.; Zenisek, K. Economical parallel oligonucleotide and peptide synthesizer - Pet Oligator. International Journal of Peptide Research and Therapeutics 2007, 13 (1-2), 367-375. 2007IntJPeptResTherap.pdf
- Raman, B.; Kotseroglou, T.; Clark, L.; Lebl, M.; Gutierrez-Osuna, R. Neuromorphic processing for optical microbead arrays: dimensionality reduction and contrast enhancement. IEEE Sensors Journal 2007, 7 (4), 506-514. 2007IEEESensorsJournal.pdf
- Shiryaev, S. A.; Kozlov, I. A.; Ratnikov, B. I.; Smith, J. W.; Lebl, M.; Strongin, A. Y. Cleavage preference distinguishes the two-component NS2B-NS3 serine proteinases of Dengue and West Nile viruses. Biochem. J. 2007, 401, 743-752. 2007BiochemJ.pdf
- Shiryaev, S. A.; Ratnikov, B. I.; Aleshin, A. E.; Kozlov, I. A.; Nelson, N. A.; Lebl, M.; Smith, J. W.; Liddington, R. C.; Strongin, A. Y. Switching the substrate specificity of the two-component NS2B-NS3 flaviviral proteinase by structure-based mutagenesis. J. Virol. 2007, 81 (9), 4501-4509. 2007JVirology.pdf
- Shiryaev, S. A.; Remacle, A. G.; Ratnikov, B. I.; Nelson, N. A.; Savinov, A. Y.; Wei, G.; Bottini, M.; Rega, M. F.; Parent, A.; Desjardins, R.; Fugere, M.; Day, R.; Sabet, M.; Pellecchia, M.; Liddington, R. C.; Smith, J. W.; Mustelin, T.; Guiney, D. G.; Lebl, M.; Strongin, A. Y. Targeting host cell furin proprotein convertases as a therapeutic strategy against bacterial toxins and viral pathogens. Journal of Biological Chemistry 2007, 282 (29), 20847-20853. 2007JBiolChem.pdf
- Shults, M. D.; Kozlov, I. A.; Nelson, N.; Kermani, B. G.; Melnyk, P. C.; Shevchenko, V.; Srinivasan, A.; Musmacker, J.; Hachmann, J. P.; Barker, D. L.; Lebl, M.; Zhao, C. A multiplexed protein kinase assay. Chembiochem 2007, 8, 933-942. 2007ChemBiochem.pdf
- Hachmann, J. P.; Lebl, M. Alternative to piperidine in Fmoc solid phase synthesis. J. Comb. Chem. 2006, 8, 149. 2006JCombChem.pdf
- Hachmann, J. P.; Lebl, M. Search for optimal coupling reagent in multiple peptide synthesizer. Biopolymers (Pept. Sci. ) 2006, 84, 340-347. 2006Biopolymers.pdf
- Hachmann, J. P.; Lebl, M. Synthesis of poly d(G-C) oligonucleotides. Nucleosides, Nucleotides and Nucleic Acids 2006, 25 (7), 705-717. 2006NuclNuclNuclAcids.pdf
- Kermani, B. G.; Fomenko, I.; Kotseroglou, T.; Forood, B.; Clark, L.; Barker, D.; Lebl, M. Decoding beads in a randomly assembled optical nose. Sensors and Actuators B 2006, 117, 282-285. 2006SensorsActuatorsB.pdf
- Kozlov, I. A.; Melnyk, P. C.; Zhao, C.; Hachmann, J. P.; Shevchenko, V.; Srinivasan, A.; Barker, D. L.; Lebl, M. A method for rapid protease substrate evaluation and optimization. Comb. Chem. High Throughput Screening 2006, 9, 481-487. 2006CombChemHighThrScr.pdf
- Lebl, M.; Barker, D. L.; Kozlov, I. A.; Melnyk, P. C.; Hachmann, J. P.; Srinivasan, A.; Shults, M.; Nelson, N.; Zhao, C. Multiplexed profiling of protease and kinase substrate with readout on oligonucleotide microarrays. J. Peptide Sci. 2006, 12, 95. WOS:000239905600053
- Lebl, M.; Hachmann, J. P. High-throughput peptide synthesis. Howl, J., Ed.; Humana Press, Inc.: Totowa, NJ, 2005; pp 167-194. 2005MethMolBiol.pdf
- Lebl, M. Combinatorial chemistry. In: Encyclopedia of 20th-Century Technology, Hempstead, C. A., Worthington, W. E., Eds.; Routledge: New York, 2005; pp 171-174. 2005Encyclopedia20thCentTechnol.pdf
- Lebl, M.; Pokorny, V.; Krchnak, V. Simple tools for resin distribution. J. Comb. Chem. 2005, 7, 42-45. 2005JCombChem.pdf
- Kermani, B.; Fomenko, I.; Kotseroglou, T.; Forood, B.; Clark, L.; Barker, D.; Lebl, M. Supervised learning for decoding beads in a randomly-assembled optical nose. In: Computational Biology Workshop, Neural Information Processing System (NIPS), 11th Annual Conference, Whistler, BC, Canada, 2004. 2002ONosePosters.pdf
- Kermani, B.; Kotseroglou, T.; Forood, B.; Barker, D.; Lebl, M. Optical nose signal denoising and detrending using wavelets. In: Proceedings of 8th World Multiconference on Systems, Cybernetics, and Informatics, Orlando, FL, 2004; pp 148-149. 2002ONosePosters.pdf
- Lebl, M. Centrifugation based automated synthesis technologies. J. Assoc. Lab. Autom. 2003, 8 (3), 30-36. 2003JALA.pdf
- Forood, B.; Kotseroglou, T.; Clark, L.; Lebl, M.; Lieu, M.-H.; Kermani, B.; Barker, D.; Dickinson, T. Chemical detection using Illumina's BeadArray technology. In: Proc. 9th International Symposium on Olfaction and Electronic Nose, ISOEN'02, Rome, 2002. 2002ONosePosters.pdf
- Lam, K. S.; Lebl, M. Synthesis of one-bead-one-compound combinatorial peptide library. In: Protein Protocols on CD-ROM Version 2.0, John M.Walker, Ed.; Humana Press: Totowa, NJ, 2002; pp 20-24. 2002ProtProtocolsCD.pdf
- Lebl, M. Combinatorial chemistry: The history and the basics. In: Integrated Drug Discovery Technologies; 2002. 2002IntegrDrugDiscTechnol.pdf
- Lebl, M.; Pires, J.; Burger, C.; Ni, Y.; Chen, Y. Solid-phase parallel synthesis of large tetrahydroisoquinolinone library. In: High-Throughput Synthesis, Sucholeiki, I., Ed.; Marcel Dekker, Inc.: New York, 2001; pp 187-195. 2001HighThrSynt_187.pdf
- Lebl, M.; Burger, C.; Ellman, B.; Heiner, D.; Ibrahim, G.; Jones, A.; Nibbe, M.; Thompson, J.; Mudra, P.; Pokorny, V.; Poncar, P.; Zenisek, K. Fully automated parallel oligonucleotide synthesizer. Collect. Czech. Chem. Commun. 2001, 66, 1299-1314. 2001CCCC.pdf
- Lebl, M.; Pires, J. Solid-phase parallel synthesis of a large array of tetrahydroisoquinolinones. In: High-Throughput Synthesis, Sucholeiki, I., Ed.; Marcel Dekker, Inc.: New York, 2001; pp 197-205. 2001HighThrSynt_197.pdf
- Lebl, M.; Houghten, R. A. Preface. In: Peptides; The Wave of the Future. Proc. 2nd Int. 17th Amer. Pept. Symp.; Lebl, M., Houghten, R. A., Eds.; American Peptide Society: San Diego, 2001; p ix-xi. 2001Proc17APS.pdf
- Lebl, M.; Burger, C.; Ellman, B.; Heiner, D.; Ibrahim, G.; Jones, A.; Nibbe, M.; Pires, J.; Mudra, P.; Pokorny, V.; Poncar, P.; Zenisek, K. Fully automated parallel oligonucleotide synthesizer. In: Peptides; The Wave of the Future. Proc. 2nd Int. 17th Amer. Pept. Symp.; Lebl, M., Houghten, R. A., Eds.; American Peptide Society: San Diego, 2001; pp 277-278. 2001Proc17APS_277.pdf
- Eichler, J.; Lebl, M. Combinatorial chemistry: A powerful tool for basic research and drug discovery. Journal of Clinical Ligand Assay 2000, 23 (4), 262-272. 2000JClinLigAssay.pdf
- Eichler, J.; Lebl, M. La chimica combinatoria: un potente strumento per la ricerca di base e la ricerca farmacologica. Journal of Clinical Ligand Assay 2000, 23, 262-272. 2000JCLA_Italian.pdf
- Lebl, M.; Ma, J.; Pires, J.; Dooley, C.; Houghten, R. A. Rapid parallel synthesis of 584 betides, peptides composed largely of beta-amino acids with side-chains not found in natural peptides. In: Peptides for the New Millennium, Fields, G. B., Tam, J. P., Barany, G., Eds.; Kluwer Academic Publisher: Dordrecht, 2000; pp 174-175. 1999Proc16APS_174.pdf
- Lebl, M. New technique for high-throughput synthesis of peptides, peptidomimetics and nonpeptide small organic molecule arrrays. In: Peptides for the New Millennium, Fields, G. B., Tam, J. P., Barany, G., Eds.; Kluwer Academic Publisher: Dordrecht, 2000; pp 164-166. 1999Proc16APS_164.pdf
- Ni, Y.; Krchnak, V.; Lebl, M. New approach for preparation of 2,3,7-trisubstituted 3,4-dihydroisoquinolinone libraries on solid phase. Mol. Diversity 2000, 5 (3), 153-161. 2000MolDiv.pdf
- Lebl, M. New approaches to automatic synthesis of large arrays of small organic molecules. In: Proceedings of combinatorial chemistry conference; Osaka, Japan, 1999; pp 6-14. 1999ProcOsaka.pdf
- Lebl, M.; Pires, J.; Poncar, P.; Pokorny, V. Evaluation of gaseous hydrogen fluoride as a convenient reagent for parallel cleavage from the solid support. J. Comb. Chem. 1999, 1 (6), 474-479. 1999JCombChem_474.pdf
- Lebl, M. Sooner or later someone else will cotton on to this idea (in " Matrix Assisted Synthetic Transformations: A Mosaic of Diverse Contributions. II. The Pattern Is Completed" by D. Hudson). J. Comb. Chem. 1999, 1 (6), 438-442. 1999JCombChem_403.pdf
- Lebl, M. New technique for high-throughput synthesis. Bioorg. Med. Chem. Lett. 1999, 9 (9), 1305-1310. 1999BioorgMedChemLett.pdf
- Lebl, M. Parallel personal comments on "classical" papers in combinatorial chemistry. J. Comb. Chem. 1999, 1 (1), 3-24. 1999JCombChem_003.pdf
- Lebl, M.; Krchnak, V.; Ibrahim, G.; Pires, J.; Burger, C.; Ni, Y.; Chen, Y.; Podue, D.; Mudra, P.; Pokorny, V.; Poncar, P.; Zenisek, K. Solid-phase synthesis of large tetrahydroisoquinolinone arrays by two different approaches. Synthesis-Stuttgart 1999, (11), 1971-1978. 1999Synthesis.pdf
- Lebl, M.; Krchnak, V. Techniques for massively parallel synthesis of small organic molecules. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1999; pp 43-46. 1998InnovPerspSPS_043.pdf
- Lebl, M. Solid-phase synthesis of combinatorial libraries. Curr. Opin. Drug. Disc. Develop. 1999, 2 (4), 385-395. 1999CurrOpinDrugDiscDev.pdf
- Rinnova, M.; Lebl, M.; Soucek, M. Solid-phase peptide synthesis by fragment condensation: Coupling in swelling volume. Lett. Peptide Sci. 1999, 6, 15-22. 1999LettPeptSci.pdf
- Rinnova, M.; Soucek, M.; Voburka, Z.; Lebl, M.; Fusek, M. Sanger's reagent: An excellent end-capping and/or labeling agent for SPPS. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1999; pp 385-386. 1998InnovPerspSPS_385.pdf
- Thorpe, D. S.; Yeoman, H.; Chan, A. W. E.; Krchnak, V.; Lebl, M.; Felder, S. Combinatorial chemistry reveals a new motif that binds the platelet fibrinogen receptor, gpIIbIIIa. Biochem. Biophys. Res. Commun. 1999, 256 (3), 537-541. 1999BiochemBiophyResComm.pdf
- Lam, K. S.; Lebl, M. Synthesis of a one-bead one-compound combinatorial peptide library. Methods in Molecular Biology (Totowa, New Jersey) 1998, 87 (Combinatorial Peptide Library Protocols), 1-6. 1998CombPeptLibProt.pdf
- Lebl, M. Solid-phase synthesis on planar supports. Biopolymers (Pept. Sci. ) 1998, 47 (5), 397-404. 1998PeptSci_397.pdf
- Lebl, M. A new approach to automated solid phase synthesis based on centrifugation of tilted plates. J. Assoc. Lab. Autom. 1998, 3 (3), 59-61. 1998JALA.pdf
- Ostrem, J. A.; Al-Obeidi, F.; Safar, P.; Safarova, A.; Stringer, S. K.; Patek, M.; Cross, M. T.; Spoonamore, J.; LoCascio, J. C.; Kasireddy, P.; Thorpe, D. S.; Sepetov, N.; Lebl, M.; Wildgoose, P.; Strop, P. Discovery of a novel, potent, and specific family of factor Xa inhibitors via combinatorial chemistry. Biochemistry 1998, 37 (4), 1053-1059. 1998Biochemistry.pdf
- Patek, M.; Lebl, M. Safety-catch and multiply cleavable linkers in solid-phase synthesis. Biopolymers (Pept. Sci. ) 1998, 47 (5), 353-363. 1998PeptSci_353.pdf
- Seligmann, B.; Lebl, M.; Lam, K. S. Solid-phase peptide synthesis, lead generation, and optimization. In: Combinatorial Chemistry and Molecular Diversity in Drug Discovery, Gordon, E. M., Kerwin, J. F. J., Eds.; John Wiley & Sons: New York, 1998; pp 39-109. 1998CombChemMolDivDrugDisc.pdf
- Cargill, J. F.; Lebl, M. New methods in combinatorial chemistry: Robotics and parallel synthesis. Curr. Opin. Chem. Biol. 1997, 1 (1), 67-71. 1997CurrOpinChemBiol.pdf
- Krchnak, V.; Weichsel, A. S.; Lebl, M.; Felder, S. Automated solid-phase organic synthesis in micro-plate wells. Synthesis of N-(alkoxy-acyl)amino alcohols. Bioorg. Med. Chem. Lett. 1997, 7 (8), 1013-1016. 1997BioorgMedChemLett.pdf
- Lam, K. S.; Lebl, M.; Krchnak, V. The "one-bead-one-compound" combinatorial library method. Chem. Rev. 1997, 97 (2), 411-448. 1997ChemRev.pdf
- Lebl, M.; Krchnak, V. Synthetic peptide libraries. Methods Enzymol. 1997, 289, 336-392. 1997MethEnzymol.pdf
- Chen, C. L.; Strop, P.; Lebl, M.; Lam, K. S. One bead-one compound combinatorial peptide library: Different types of screening. Methods Enzymol. 1996, 267, 211-219. 1996MethEnzymol.pdf
- Eichler, J.; Houghten, R. A.; Lebl, M. Inclusion volume solid-phase peptide synthesis. J. Peptide Sci. 1996, 2 (4), 240-244. 1996JPeptSci.pdf
- Hruby, V. J.; Shenderovich, M.; Lam, K. S.; Lebl, M. Design considerations and computer modeling related to the development of molecular scaffolds and peptide mimetics for combinatorial chemistry. Mol. Diversity 1996, 2 (1-2), 46-56. 1996MolDiv_46.pdf
- Krchnak, V.; Weichsel, A. S.; Cabel, D.; Lebl, M. Structurally homogenous and heterogenous libraries: Scaffold- based libraries and libraries built using bifunctional building blocks. In: Molecular Diversity and Combinatorial Chemistry. Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; American Chemical Society: Washington,DC, 1996; pp 99-117. 1996MolDivCombChem.pdf
- Krchnak, V.; Vagner, J.; Flegelova, Z.; Weichsel, A. S.; Barany, G.; Lebl, M. Use of solid-phase Mitsunobu and Wittig reactions for contruction of peptide and non-peptide libraries. In: Peptides:Chemistry,Structure and Biology,Proc.14.APS, Kaumaya, P. T. P., Hodges, R. S., Eds.; Mayflower Scientific Ltd.: Kingswinford, 1996; pp 307-308. 1996Proc14APS_307.pdf
- Krchnak, V.; Lebl, M. MARS: Multiple automatic robot synthesizer featuring a novel timing procedure and random access to reagents and reaction vessels. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1996; pp 93-96. 1996InnovPerspSPS_093.pdf
- Krchnak, V.; Sepetov, N. F.; Kocis, P.; Patek, M.; Lam, K. S.; Lebl, M. Combinatorial libraries of synthetic structures: Synthesis, screening, and structure determination. In: Combinatorial Libraries: Synthesis, Screening and Application Potential, Cortese, R., Ed.; Walter de Gruyter: Berlin, 1996; pp 27-52. 1996CombLib_Cortese.pdf
- Krchnak, V.; Weichsel, A. S.; Cabel, D.; Flegelova, Z.; Lebl, M. Structurally homogenous and heterogenous synthetic combinatorial libraries. Mol. Diversity 1996, 1 (3), 149-164. 1995MolDiv_149.pdf
- Krchnak, V.; Lebl, M. Synthetic library techniques: Subjective (biased and generic) thoughts and views. Mol. Diversity 1996, 1 (3), 193-216. 1995MolDiv_193.pdf
- Krchnak, V.; Cabel, D.; Lebl, M. MARS: Multiple automated robotic synthesizer for continuous flow of peptides. Peptide Res. 1996, 9 (1), 45-49. 1996PeptRes_45.pdf
- Lam, K. S.; Lou, Q.; Zhao, Z. G.; Chen, M. L.; Salmon, S. E.; Wade, S.; Lebl, M. Identification and applications of idiotype-specific peptides for two murine B-cell lymphoma cell lines. In: Peptides:Chemistry,Structure and Biology,Proc.14.APS, Kaumaya, P. T. P., Hodges, R. S., Eds.; Mayflower Scientific Ltd.: Kingswinford, 1996; pp 806-807. 1996Proc14APS_806.pdf
- Lam, K. S.; Lebl, M. Combinatorial library based on the one-bead-one-compound concept. In: Combinatorial Peptide and Nonpeptide Libraries: A Handbook, Jung, G., Ed.; VCH: Weinheim, 1996; pp 173-201. 1996CombPeptNonpeptLibraries.pdf
- Lam, K. S.; Lake, D.; Salmon, S. E.; Smith, J.; Chen, M. L.; Wade, S.; Abdul-Latif, F.; Leblova, Z.; Ferguson, R. D.; Krchnak, V.; Sepetov, N. F.; Lebl, M. A one-bead one-peptide combinatorial library method for B-cell epitope mapping. Methods: A Companion to Methods in Enzymology 1996, 9, 482-493. 1996Methods_482.pdf
- Lebl, M.; Krchnak, V.; Strop, P.; Lam, K. S. Construction and screening of peptide and nonpeptide libraries based on one-bead-one-compound principle. In: Peptides:Chemistry,Structure and Biology,Proc.14.APS, Kaumaya, P. T. P., Hodges, R. S., Eds.; Mayflower Scientific Ltd.: Kingswinford, 1996; pp 890-892. 1996Proc14APS_890.pdf
- Lebl, M.; Krchnak, V.; Patek, M.; Lam, K. S. Synthetic combinatorial libraries of scaffolded and unordered structures. Methods Mol. Cell. Biol. 1996, 6 (1), 41-55. 1995MethMolCellBiol_41.pdf
- Rinnova, M.; Fusek, M.; Lebl, M. Use of methyl red in solid phase synthesis. In: Innovation and Perspectives in Solid Phase Synthesis & Combinatorial Libraries, Epton, R., Ed.; Mayflower Scientific Limited: Birmingham, 1996; pp 509-510. 1996InnovPerspSPS_509.pdf
- Rinnova, M.; Lebl, M. Molecular diversity and libraries of structures: Synthesis and screening. Collect. Czech. Chem. Commun. 1996, 61, 171-231. 1996CCCC_0171.pdf
- Salmon, S. E.; Liu-Stevens, R. H.; Zhao, Y.; Lebl, M.; Krchnak, V.; Wertman, K.; Sepetov, N.; Lam, K. S. High-volume cellular screening for anticancer agents with combinatorial chemical libraries: A new methodology. Mol. Diversity 1996, 2 (1-2), 57-63. 1996MolDiv_57.pdf
- Stankova, M.; Lebl, M. Library generation through successive substitution of trichlorotriazine. Mol. Diversity 1996, 2 (1-2), 75-80. 1996MolDiv_75.pdf
- Stankova, M.; Strop, P.; Chen, C.; Lebl, M. Mixtures of molecules versus mixtures of pure compounds on polymeric beads. In: Molecular Diversity and Combinatorial Chemistry. Libraries and Drug Discovery, Chaiken, I. M., Janda, K. D., Eds.; American Chemical Society: Washington,DC, 1996; pp 137-143. 1996MolDivCombChem.pdf
- Vagner, J.; Krchnak, V.; Lebl, M.; Barany, G. Solid-phase organic synthesis: Creation of carbon-carbon double bond under mild conditions by Wittig-type reactions. Collect. Czech. Chem. Commun. 1996, 61, 1697-1702. 1996CCCC_1697.pdf
- Vagner, J.; Barany, G.; Lam, K. S.; Krchnak, V.; Sepetov, N. F.; Ostrem, J. A.; Strop, P.; Lebl, M. Enzyme-mediated spatial segregation on individual polymeric support beads: Application to generation and screening of encoded combinatorial libraries. Proc. Natl. Acad. Sci. USA 1996, 93 (16), 8194-8199. 1996PNAS_Vagner.pdf
- Flegelova, Z.; Krchnak, V.; Sepetov, N. F.; Stankova, M.; Issakova, O.; Cabel, D.; Lam, K. S.; Lebl, M. Libraries of small compact structures based on N-acyl-N-alkylamino acids. In: Peptides 94, Proc.23.EPS, Maia, H. L. S., Ed.; ESCOM: Leiden, 1995; pp 469-470. 1995Proc23EPS_469.pdf
- Geysen, H. M.; Houghten, R. A.; Kauffman, S.; Lebl, M.; Moos, W. H.; Pavia, M. R.; Szostak, J. W. Molecular diversity comes of age. Mol. Diversity 1995, 1 (1), 1-3. 1995MolDiv_001.pdf
- Kasal, A.; Kohout, L.; Lebl, M. Synthesis of a scaffold for the creation of non-peptide libraries. Collect. Czech. Chem. Commun. 1995, 60, 2147-2155. 1995CCCC_2147.pdf
- Kocis, P.; Issakova, O.; Sepetov, N. F.; Lebl, M. Kemp's triacid scaffolding for synthesis of combinatorial nonpeptide uncoded libraries. Tetrahedron Lett. 1995, 36, 6623-6626. 1995TetLett_6623.pdf
- Krchnak, V.; Weichsel, A. S.; Cabel, D.; Lebl, M. Linear presentation of variable side-chain spacing in a highly diverse combinatorial library. Peptide Res. 1995, 8 (4), 198-205. 1995PeptRes_198.pdf
- Krchnak, V.; Weichsel, A. S.; Issakova, O.; Lam, K. S.; Lebl, M. Bifunctional scaffolds as templates for synthetic combinatorial libraries. Mol. Diversity 1995, 1 (3), 177-182. 1995MolDiv_177.pdf
- Krchnak, V.; Flegelova, Z.; Weichsel, A. S.; Lebl, M. Polymer-supported Mitsunobu ether formation and its use in combinatorial chemistry. Tetrahedron Lett. 1995, 36, 6193-6196. 1995TetLett_6193.pdf
- Lam, K. S.; Lebl, M.; Wu, J.; Wade, S.; Lou, Q.; Zhao, Z. G.; Chen, M. L.; Chang, M. P.; Smith, M.; Grimes, W. J. Peptide library screening based on the one-bead one-peptide concept: An update. In: Peptides 94, Proc.23.EPS, Maia, H. L. S., Ed.; ESCOM: Leiden, 1995; pp 453-454. 1995Proc23EPS_453.pdf
- Lam, K. S.; Lebl, M. Synthesis and screening of a "one-bead-one-compound" combinatorial peptide library. Methods Mol. Cell. Biol. 1995, 6 (1), 15-25. 1995MethMolCellBiol_15.pdf
- Lam, K. S.; Lebl, M. Peptide library screening based on the one-bead-one-peptide concept. In: Peptides:Biology and Chemistry,Proc.1994 Chinese Peptide Symposium, Lu, G. S., Tam, J. P., Du, Y. C., Eds.; ESCOM: Leiden, 1995; pp 273-277. 1994ProcCPS_273.pdf
- Lam, K. S.; Wade, S.; Abdul-Latif, F.; Lebl, M. Application of a dual color detection scheme in the screening of a random combinatorial peptide library. J. Immunol. Method 1995, 180 (2), 219-223. 1995JImmunolMeth.pdf
- Lebl, M.; Krchnak, V.; Sepetov, N. F.; Seligmann, B.; Strop, P.; Felder, S.; Lam, K. S. One-bead-one-structure combinatorial libraries. Biopolymers (Pept. Sci. ) 1995, 37 (3), 177-198. 1995PeptSci_177.pdf
- Lebl, M.; Krchnak, V.; Sepetov, N. F.; Nikolaev, V.; Stankova, M.; Kocis, P.; Patek, M.; Flegelova, Z.; Ferguson, R.; Lam, K. S. Synthetic combinatorial libraries: A new tool for drug design. Methods for identifying the composition of compounds from peptide and/or nonpeptide libraries. In: Methods in Protein Structure Analysis, Atassi, M. Z., Appella, E., Eds.; Plenum Press: New York, 1995; pp 335-342. 1995MethProtStrAnal.pdf
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- Krchnak, V.; Vagner, J.; Eichler, J.; Lebl, M. Color monitored solid phase peptide synthesis. In: Peptides 1988,Proc.20.EPS, Jung, G., Bayer, E., Eds.; Walter de Gruyter & Co.: Berlin, 1989; pp 232-234. 1989Proc20EPS_232.pdf
- Lebl, M.; Barth, T.; Slaninova, J.; Hrbas, P.; Eichler, J.; Cerny, B. Synthesis, tritiation and biological studies with [2-O-methyltyrosine, 7-(3,4-dehydroproline)]deamino-1-carba-oxytocin. In: Peptides 1988,Proc.20.EPS, Jung, G., Bayer, E., Eds.; Walter de Gruyter & Co.: Berlin, 1989; pp 546-548. 1989Proc20EPS_546.pdf
- Lebl, M.; Slaninova, J.; Johnson, R. L. Analogs of oxytocin containing a pseudopeptide Leu-Gly bond of cis and trans configuration. Int. J. Peptide Prot. Res. 1989, 33, 16-21. 1989IntJPeptProtRes_16.pdf
- Lebl, M.; Hruby, V. J.; Castrucci, A. M. L.; Hadley, M. E. Melanin concentrating hormone analogues: Contraction of the cyclic structure. II.Antagonist activity. Life Sci. 1989, 44 (7), 451-457. 1989LifeSci_0451.pdf
- Lebl, M.; Eichler, J. Simulation of continuous solid phase synthesis: Synthesis of methionine enkephalin and its analogs. Peptide Res. 1989, 2 (4), 297-300. 1989PeptRes_297.pdf
- Matsunaga, T. O.; Hruby, V. J.; Lebl, M.; Castrucci, A. M. L.; Hadley, M. E. Melanin concentrating hormone (MCH): Structure-function aspects of its melanocyte stimulating hormone-like (MSH-like) activity. Peptides 1989, 10, 773-778. 1989Peptides.pdf
- Slaninova, J.; Lebl, M.; Eichler, J. Synthesis and properties of antiparallel dimer of deamino-1-carba-oxytocin. In: Peptides 1988,Proc.20.EPS, Jung, G., Bayer, E., Eds.; Walter de Gruyter & Co.: Berlin, 1989; pp 543-545. 1989Proc20EPS_543.pdf
- Zicha, J.; Kunes, J.; Lebl, M.; Pohlova, I.; Slaninova, J.; Jelinek, J. Antidiuretic and pressor actions of vasopressin in age-dependent DOCA-salt hypertension. Amer. J. Physiol. 1989, 256 (1;Part 2), R138-R145. 1989AmJPhysiol.pdf
- Bendlova, B.; Lebl, M.; Stolba, P.; Starka, L. Synthesis of modified human C-peptide and its fragments. Collect. Czech. Chem. Commun. 1988, 53, 2637-2644. 1988CCCC_2637.pdf
- Fassina, G.; Lebl, M.; Chaiken, I. Screening the recognition properties of peptide hormone sequence mutants by analytical high performance liquid affinity chromatography on immobilized neurophysin. Collect. Czech. Chem. Commun. 1988, 53, 2627-2636. 1988CCCC_2627.pdf
- Krchnak, V.; Vagner, J.; Safar, P.; Lebl, M. Noninvasive continuous monitoring of solid phase peptide synthesis by acid-base indicator. Collect. Czech. Chem. Commun. 1988, 53, 2542-2548. 1988CCCC_2542.pdf
- Krchnak, V.; Vagner, J.; Lebl, M. Noninvasive continuous monitoring of solid phase peptide synthesis by acid-base indicator (preliminary communication). Int. J. Peptide Prot. Res. 1988, 32 (5), 415-416. 1988IntJPeptProtRes_415.pdf
- Lebl, M.; Hruby, V. J.; Castrucci, A. M. L.; Visconti, M. A.; Hadley, M. E. Melanin concentrating hormone analogues: Contraction of the cyclic structure. 1.Agonist activity. J. Med. Chem. 1988, 31 (5), 949-954. 1988JMedChem.pdf
- Mader, P.; Vesela, V.; Heyrovsky, M.; Lebl, M.; Braunsteinova, M. Polarography of the oxytocin and vasopressin synthetic analogs. Collect. Czech. Chem. Commun. 1988, 53, 1579-1605. 1988CCCC_1579.pdf
- Prochazka, Z.; Ancans, J. E.; Slaninova, J.; Machova, A.; Barth, T.; Skopkova, J.; Budesinsky, M.; Pavlikova, F.; Lebl, M. Synthesis and properties of analogues of vasopressin with 1-aminocyclopropane-1-carboxylic acid. Collect. Czech. Chem. Commun. 1988, 53, 2604-2616. 1988CCCC_2604.pdf
- Barth, T.; Slaninova, J.; Lebl, M.; Hruby, V. J. Effect of threonine in position 4 in oxytocin and vasotocin analogs on the time course of uterotonic response. Endocrinol. Exper. 1987, 21 (3), 191-197. 1987EndocrinolExper.pdf
- Hruby, V. J.; Lebl, M. Conformational properties of neurohypophyseal hormone analogs in solution as determined by NMR and laser Raman spectroscopies. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 105-155.
- Jost, K.; Lebl, M.; Brtnik, F. Nomenclature. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 5-8.
- Jost, K.; Lebl, M.; Brtnik, F. Introductory remarks. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 1-4.
- Lebl, M. Analogs with dissociated and/or high activities. II.Uterotonic activity. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 78-102.
- Lebl, M.; Jost, K.; Brtnik, F. Tables of analogs. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 127-268.
- Lebl, M.; Sugg, E. E.; Van Binst, G.; van der Elst, P.; Tourwe, D.; Slaninova, J.; Hruby, V. J. Analogs of oxytocin containing a modified peptide bond. Int. J. Peptide Prot. Res. 1987, 30 (3), 318-322. 1987IntJPeptProtRes_318.pdf
- Lebl, M. Analogs with dissociated and/or high activities. III. Galactogogic activity. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 102-109.
- Lebl, M. Analogs with dissociated and/or high activities. I.Introduction. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 75-78.
- Lebl, M. Synthesis, purification, and stability of the neurohypophyseal hormone analogs. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 23-82.
- Lebl, M. Modification of other functional groups. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 156-160.
- Lebl, M. Isotopically modified analogs. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 83-104.
- Lebl, M.; Sugg, E. E.; Hruby, V. J. Proton NMR spectroscopic evidence for sulfur-aromatic interactions in peptides. Int. J. Peptide Prot. Res. 1987, 29 (1), 40-45. 1987IntJPeptProtRes_040.pdf
- Lebl, M. Analogs with inhibitory properties. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 17-74.
- Lebl, M.; Hruby, V. J. Other methods used in the investigation of neurohypophyseal hormone analog conformations. In: CRC Handbook of Neurohypophyseal Hormone Analogs, Jost, K., Lebl, M., Brtnik, F., Eds.; CRC Press: Boca Raton, 1987; pp 155-159.
- Lebl, M.; Fric, I.; Sugg, E. E.; Cody, W. L.; Hruby, V. J. Conformational studies of carba-analogs of oxytocin. In: Peptides 1986, Proc.19.EPS, Theodoropoulos, D., Ed.; Walter de Gruyter & Co.: Berlin, 1987; pp 341-344. 1986Proc19EPS_341.pdf
- Zaoral, M.; Blaha, I.; Lebl, M.; Barth, T. Vasopressin analogs with strong agonistic-antagonistic properties. In: Peptides 1986, Proc.19.EPS, Theodoropoulos, D., Ed.; Walter de Gruyter & Co.: Berlin, 1987; pp 465-468. 1986Proc19EPS_465.pdf
- Zicha, J.; Kunes, J.; Lebl, M.; Pohlova, I.; Jelinek, J. Haemodynamics and the participation of pressor systems in young and adult rats with age-dependent doca-salt hypertension. Physiol. Bohemoslov. 1987, 36, 89-92. 1987PhysiolBohem.pdf
- Hermann, P.; Jannasch, R.; Lebl, M. Application of high-performance liquid chromatography and capillary isotachophoresis to the purification and characterization of products of peptide synthesis. J. Chromatogr. 1986, 351, 283-293. 1986JChromatogr.pdf
- Hrbas, P.; Barth, T.; Lebl, M.; Papsuevich, A. O.; Flegel, M. Mono- and diiodo-derivatives of neurohypophysial hormones and their analogues. Beitr. Wirkstofforsch. 1985, 24, 182-187. 1985BeitrWirkst.pdf
- Lebl, M.; Drasar, P.; Koroniak, H.; Milecki, J.; Ikonomov, O. C. Nejnovejsí poznatky v chemii porkanovych sloucenin. Chem. Listy 1985, 79, 410-417. 1985ChemListy.pdf
- Lebl, M. Carba analogues of neurohypophysial hormones. In: Handbook of the Use of High Performance Liquid Chromatography for the Analytical and Preparative Separation of Amino Acids, Peptides and Proteins, Hancock, W. S., Ed.; CRC Press: Boca Raton, 1985; pp 169-178. 1985HandbookHPLC.pdf
- Lebl, M.; Barth, T.; Servitova, L.; Slaninova, J.; Jost, K. Oxytocin analogues with inhibitory properties, containing in position 2 a hydrophobic amino acid of D-configuration. Collect. Czech. Chem. Commun. 1985, 50, 132-145. 1985CCCC_0132.pdf
- Lebl, M.; Hruby, V. J.; Slaninova, J.; Barth, T. Solid phase synthesis and biological activities of oxytocin carba analogues containing threonine in position 4. Collect. Czech. Chem. Commun. 1985, 50, 418-427. 1985CCCC_0418.pdf
- Hrbas, P.; Skopkova, J.; Zicha, J.; Barth, T.; Lebl, M.; Jost, K. Nacartocin - analogue of oxytocin with enhanced natriuretic properties: natriuretic and hemodynamic characteristics. Endocrinol. Exper. 1984, 18 (2), 117-124. 1984EndocrinolExper.pdf
- Lebl, M.; Cody, W. L.; Wilkes, B. C.; Hruby, V. J.; Castrucci, A. M. L.; Hadley, M. E. Modification of the disulfide bridge in cyclic melanotropins. Collect. Czech. Chem. Commun. 1984, 49, 2680-2688. 1984CCCC_2680.pdf
- Lebl, M.; Cody, W. L.; Hruby, V. J. Cyclic melanotropins. Part VI. Reverse phase HPLC studies. J. Liq. Chromatogr. 1984, 7, 1195-1210. 1984JLiqChrom.pdf
- Lebl, M.; Barth, T.; Crankshaw, D. J.; Cerny, B.; Daniel, E. E.; Grover, A. K.; Jost, K. Synthesis and properties of [2-[3,5-(3)H2]-tyrosine,4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun. 1984, 49, 1921-1926. 1984CCCC_1921.pdf
- Lebl, M.; Hruby, V. J. Synthesis of cyclic peptides by solid phase technology. Tetrahedron Lett. 1984, 25 (20), 2067-2068. TetLett1984.pdf
- Lebl, M.; Barth, T.; Servitova, L.; Slaninova, J.; Hrbas, P. Synthesis and properties of carba-6-analogues of oxytocin containing a deaminopenicillamine residue in position 1. Collect. Czech. Chem. Commun. 1984, 49, 2012-2023. 1984CCCC_2012.pdf
- Lebl, M.; Cody, W. L.; Wilkes, B. C.; Hruby, V. J.; Castrucci, A. M. L.; Hadley, M. E. Cyclic melanotropins. Part VII: Modified ring structures: Synthesis and biological activity. Int. J. Peptide Prot. Res. 1984, 24 (5), 472-479. 1984IntJPeptProtRes_472.pdf
- Prochazka, Z.; Lebl, M.; Barth, T.; Hlavacek, J.; Trka, A.; Budesinsky, M.; Jost, K. Synthesis and properties of oxytocin analogues modified in the tripeptide side chain. Collect. Czech. Chem. Commun. 1984, 49, 642-652. 1984CCCC_0642.pdf
- Skopkova, J.; Barth, T.; Hrbas, P.; Jost, K.; Lebl, M. Natriuretic properties of [2-p-ethylphenylalanine]deamino-6- carba-oxytocin (Nacartocin) in cats. Exp. Clin. Endocrinol. 1984, 84, 235-238. 1984ExpClinEndocrinol.pdf
- Barth, T.; Lebl, M.; Jost, K.; Cantau, B.; Butlan, D.; Guillon, G.; Jard, S. Interactions of deamino-6-carba-oxytocin analogues in rat kidney and liver membrane systems. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 467-470. 1983Proc17EPS_467.pdf
- Barth, T.; Cantau, B.; Butlen, D.; Guillon, G.; Jard, S.; Lebl, M.; Jost, K. Oxytocin and vasopressin analogues capable of competition with vasopressin binding to rat liver membranes. Collect. Czech. Chem. Commun. 1983, 48, 1788-1795. 1983CCCC_1788.pdf
- Budesinsky, M.; Jezek, J.; Krchnak, V.; Lebl, M.; Zaoral, M.; Rotta, J.; Straka, R. Synthetic fragments of bacterial cell walls. Physicochemical and biological properties. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 305-310. 1983Proc17EPS_305.pdf
- Butlen, D.; Barth, T.; Cantau, B.; Guillon, G.; Jard, S.; Lebl, M.; Brtnik, F.; Jost, K. The structural requirements of oxytocin and vasopressin analogues for the activation of adenylate cyclase in the rat kidney medullary membrane system. Collect. Czech. Chem. Commun. 1983, 48, 3166-3176. 1983CCCC_3166.pdf
- Krojidlo, M.; Flegel, M.; Lebl, M. Method for cyclization of carba analogues of oxytocin. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 199-202. 1983Proc17EPS_199.pdf
- Lebl, M.; Barth, T.; Servitova, L.; Slaninova, J.; Jost, K. Analogues of neurohypophysial hormones containing a D-amino acid in position 2. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 457-460. 1983Proc17EPS_457.pdf
- Lebl, M. Analogues of neurohypophysial hormones with inhibitory effect on the pressoric activity of vasopressin. In: Vasopressin and Pathology of the Cardiovascular System in Aging, Chebotarev, D. F., Frolkis, V. V., Eds.; Institute of Gerontology: Kiev, 1983; pp 108-114. 1983VasopPathCardioSystAging.pdf
- Lebl, M.; Barth, T. Synthesis and some activities of [1-penicillamine]deamino-6-carba-oxytocin. In: Peptides:Structure and Function,Proc.8.APS, Hruby, V. J., Rich, D. H., Eds.; Pierce: Rockford, 1983; pp 357-360. 1983Proc8APS_357.pdf
- Lebl, M.; Gut, V. Calculation of the rate constant of a reversible reaction from the chromatographic peaks for muranyl dipeptide anomers. J. Chromatogr. 1983, 260, 478-482. JChromatogr1983_Gut.pdf
- Lebl, M. Amino acids and peptides CLXXXI. Separation of diastereoisomers of oxytocin analogues. J. Chromatogr. 1983, 264, 459-462. 1983JChromatogr_459.pdf
- Prochazka, Z.; Lebl, M.; Barth, T.; Hlavacek, J.; Jost, K. Two analogues of oxytocin with modified proline cyclic structure. In: Peptides 1982,Proc.17.EPS, Blaha, K., Malon, P., Eds.; Walter de Gruyter: Berlin, 1983; pp 441-444. 1983Proc17EPS_441.pdf
- Lebl, M.; Pospisek, J.; Hlavacek, J.; Barth, T.; Malon, P.; Servitova, L.; Hauzer, K.; Jost, K. Analogues of neurohypophysial hormones containing tert.leucine: synthesis and properties. Collect. Czech. Chem. Commun. 1982, 47, 689-701. 1982CCCC_0689.pdf
- Lebl, M. Correlation between hydrophobicity of substituents in the phenylalanine moiety of oxytocin carba-analogues and reversed- phase-chromatographic k' values. J. Chromatogr. 1982, 242, 342-345. 1982JChromatogr.pdf
- Lebl, M.; Hrbas, P.; Skopkova, J.; Slaninova, J.; Machova, A.; Barth, T.; Jost, K. Synthesis and properties of oxytocin analogues with high and selective natriuretic activity. Collect. Czech. Chem. Commun. 1982, 47, 2540-2560. 1982CCCC_2540.pdf
- Barth, T.; Hrbas, P.; Skopkova, J.; Slaninova, J.; Lebl, M.; Jost, K. Natriuretic effects of oxytocin analogues. In: Peptides 1980,Proc.16.EPS, Brunfeldt, K., Ed.; Scriptor: Copenhagen, 1981; pp 416-419. 1981Proc16EPS_416.pdf
- Barth, T.; Slaninova, J.; Servitova, L.; Lebl, M.; Kotsira-Engonopoulos, C.; Tzougraki, C.; Photaki, I.; Krojidlo, M.; Jost, K. The effect of some structural modification of the oxytocin molecule on the duration of the galactogogic response. Collect. Czech. Chem. Commun. 1981, 46, 2441-2445. 1981CCCC_2441.pdf
- Bienert, M.; Lebl, M.; Mehlis, B.; Niedrich, H. Synthesis and application of methionin S-tert-butylsulfonium peptides. In: Peptides 1980,Proc.16.EPS, Brunfeldt, K., Ed.; Scriptor: Copenhagen, 1981; pp 127-132. 1981Proc16EPS_127.pdf
- Lebl, M.; Barth, T.; Jost, K. Chromatographic and pharmacological properties of carba- analogues of neurohypophyseal hormones sulfoxides. A general method of sulfoxide group determination in peptides. In: Peptides 1980,Proc.16.EPS, Brunfeldt, K., Ed.; Scriptor: Copenhagen, 1981; pp 719-724. 1981Proc16EPS_719.pdf
- Prochazka, Z.; Lebl, M.; Servitova, L.; Barth, T.; Jost, K. Synthesis and pharmacological properties of 2-p-fluorophenyl- alanine deamino-1-carba-oxytocin and of its diastereoisomeric sulfoxides. Collect. Czech. Chem. Commun. 1981, 46, 947-956. 1981CCCC_0947.pdf
- Slaninova, J.; Lebl, M.; Barth, T.; Jost, K. The effect of magnesium ions on the uterotonic activity of carba analogues of oxytocin modified in position 4. Collect. Czech. Chem. Commun. 1981, 46, 1689-1692. 1981CCCC_1689.pdf
- Barth, T.; Slaninova, J.; Lebl, M.; Jost, K. Biological activities and protracted action of carba-analogues of deamino-oxytocin with O-methyltyrosine in position 2. Collect. Czech. Chem. Commun. 1980, 45, 3045-3050. 1980CCCC_3045.pdf
- Hrbas, P.; Barth, T.; Skopkova, J.; Lebl, M.; Jost, K. Effect of some oxytocin analogues on natriuresis in rats. Endocrinol. Exper. 1980, 14 (2), 151-157. 1980EndocrinolExper.pdf
- Hrbas, P.; Skopkova, J.; Barth, T.; Lebl, M.; Jost, K. Renal sodium excretion in rats. Effect of amino acid replacement in position 4 of the oxytocin molecule. In: Hormonal Regulation of Sodium Excretion, Lichardus, B., Schrier, R. W., Ponec, J., Eds.; Elsevier: Amsterdam, 1980; pp 169-172. 1980HormRegSodExcr_169.pdf
- Lebl, M. High-performance liquid chromatography of carba analogues of oxytocin; a method for the determination of sulfides and sulfoxides in peptides. Collect. Czech. Chem. Commun. 1980, 45, 2927-2937. 1980CCCC_2927.pdf
- Lebl, M.; Machova, A.; Hrbas, P.; Barth, T.; Jost, K. Analogues of deamino-1-carba-oxytocin with aliphatic amino acid in position 4: Chemical synthesis and biological activities. Collect. Czech. Chem. Commun. 1980, 45, 2714-2723. 1980CCCC_2714.pdf
- Lebl, M.; Barth, T.; Skopkova, J.; Jost, K. Synthesis and some pharmacological properties of [7-glycine,8- ornithine]-vasopressin and of its two analogues. Collect. Czech. Chem. Commun. 1980, 45, 2865-2871. 1980CCCC_2865.pdf
- Lebl, M.; Barth, T.; Jost, K. Synthesis and pharmacological properties of oxytocin analogues modified simultaneously in position 2 and in the disulfide bridge. Collect. Czech. Chem. Commun. 1980, 45, 2855-2864. 1980CCCC_2855.pdf
- Skopkova, J.; Hrbas, P.; Barth, T.; Lebl, M.; Jost, K. Renal sodium excretion in rats. Effect of structural modification of position 2 of deamino-6-carba-oxytocin. In: Hormonal Regulation of Sodium Secretion, Lichardus, B., Schrier, R. W., Ponec, J., Eds.; Elsevier: Amsterdam, 1980; pp 163-168. 1980HormRegSodExcr_163.pdf
- Barth, T.; Lebl, M.; Bojanovska, V.; Jost, K. Analogues of oxytocin acting as irreversible inhibitors of oxytocin. In: Peptides 1978,Proc.15.EPS, Siemion, I. Z., Kupryszewski, G., Eds.; Wroclaw University Press: Wroclaw, 1979; pp 475-479. 1979Proc15EPS_475.pdf
- Lebl, M.; Dimeli, A.; Bojanovska, V.; Slaninova, J.; Barth, T.; Jost, K. Synthesis and some biological properties of amides derived from [4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun. 1979, 44, 2556-2562. 1979CCCC_2556.pdf
- Lebl, M.; Bojanovska, V.; Barth, T.; Jost, K. Synthesis and properties of oxytocin analogues acting as irreversible inhibitors of the uterotonic response to oxytocin. Collect. Czech. Chem. Commun. 1979, 44, 2573-2582. 1979CCCC_2573.pdf
- Lebl, M.; Barth, T.; Jost, K. Analogues of oxytocin with esters of glutamic acid instead of glutamine in position 4: synthesis of a compound with high and specific galactogogic activity. Collect. Czech. Chem. Commun. 1979, 44, 2563-2572. 1979CCCC_2563.pdf
- Lebl, M.; Jost, K. Selective oxidation of sulfur in peptide synthesis. In: Peptides 1978,Proc.15.EPS, Siemion, I. Z., Kupryszewski, G., Eds.; Wroclaw University Press: Wroclaw, 1979; pp 109-112. 1979Proc15EPS_109.pdf
- Lebl, M.; Barth, T.; Jost, K. Synthesis, reduction, and pharmacological properties of the sulfoxides of some carba-analogues of oxytocin. Collect. Czech. Chem. Commun. 1978, 43, 1538-1556. 1978CCCC_1538.pdf
- Lebl, M.; Jost, K. Mechanismus racemisace derivátu aminokyselin. Chem. Listy 1978, 72, 252-266. 1978ChemListy.pdf
- Lebl, M.; Jost, K. Synthesis of [4-glutamic acid]deamino-1-carba-oxytocin. Collect. Czech. Chem. Commun. 1978, 43, 523-534. 1978CCCC_0523.pdf
- Lebl, M.; Barth, T.; Jost, K. Na-glycyl-glycyl-glycyl-8-ornithine-vasopressin: A trypsin resistant vasopressin analog with a specific pressor effect. Collect. Czech. Chem. Commun. 1978, 43, 1300-1305. 1978CCCC_1300.pdf
- Lebl, M.; Bojanovska, V.; Barth, T.; Jost, K. Oxytocin analogs effective as noncompetitive inhibitors in uterotonic test. Experientia 1978, 34 (12), 1543-1544. 1978Experientia.pdf
- Ferles, M.; Kocian, O.; Lebl, M.; Lovy, J.; Radl, S.; Silhankova, A.; Stern, P. Electrolytic reduction of quarternary salts of some alcohols of pyridine series, of corresponding alkylpyridines and alkenylpyridines. Collect. Czech. Chem. Commun. 1976, 41, 598-603. 1975CCCC_0598.pdf
- Ferles, M.; Lebl, M.; Silhankova, A.; Stern, P.; Wimmer, Z. Reduction of tertiary alcohols of the pyridine series and corresponding alkenylpyridines with zinc and formic acid. Collect. Czech. Chem. Commun. 1975, 40, 1571-1575. 1975CCCC_1571.pdf
- Ferles, M.; Lebl, M.; Stern, P.; Trska, P. Mixed electrolytic reduction of 1,4,-dimethylpyridinium methylsulfate with acetone and of 1-methylpyridinium methylsulfate with cyclopentanone. Collect. Czech. Chem. Commun. 1975, 40, 2183-2190. 1975CCCC_2183.pdf
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